SCHEMBL9765712

SCHEMBL9765712

CC1=C(C(=O)O)C(c2ccccc2Cl)C(S(=O)(=O)c2ccccc2)=C(C)N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
CYP3A4 P08684 3/20 0.40
NR1I2 O75469 2/20 0.40
TSHR P16473 4/20 0.39
POLB P06746 1/20 0.39
HSD17B10 Q99714 5/20 0.39
HPGD P15428 3/20 0.39
KDM4E B2RXH2 3/20 0.39
CASP1 P29466 3/20 0.39
CASP7 P55210 3/20 0.39
GAA P10253 2/20 0.39
GLA P06280 1/20 0.39
MAPT P10636 3/20 0.38
ALOX15 P16050 2/20 0.38
CYP2C9 P11712 3/20 0.38
TBXA2R P21731 3/20 0.38
ADRA1A P35348 3/20 0.38
SLC6A3 Q01959 3/20 0.38
MEN1 O00255 2/20 0.38
CYP1A2 P05177 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7384442 0.88 KDM4E (0.53) ALDH1A1CYP3A4NR1I2TSHRHSD17B10
SCHEMBL7272409 0.87 ALDH1A1 (0.43) ALDH1A1CYP3A4NR1I2TSHRPOLB
SCHEMBL3034308 0.85 ALDH1A1 (0.49) ALDH1A1CYP3A4NR1I2TSHRPOLB
SCHEMBL7267559 0.85 TSHR (0.44) ALDH1A1CYP3A4NR1I2TSHRPOLB
SCHEMBL7275653 0.84 ALOX15 (0.41) ALDH1A1CYP3A4NR1I2TSHRPOLB
SCHEMBL9765752 0.83 CYP3A4 (0.51) ALDH1A1CYP3A4NR1I2TSHRPOLB
SCHEMBL11362637 0.83 ALDH1A1 (0.38) ALDH1A1CYP3A4NR1I2TSHRPOLB
SCHEMBL9765774 0.81 CYP2C9 (0.46) ALDH1A1CYP3A4NR1I2TSHRHSD17B10
SCHEMBL7377019 0.80 KDM4E (0.50) ALDH1A1CYP3A4NR1I2TSHRHSD17B10
SCHEMBL7375002 0.79 KDM4E (0.49) ALDH1A1CYP3A4NR1I2TSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed