SCHEMBL9765843

SCHEMBL9765843

N#Cc1cncc(C(F)(F)F)c1.O=c1cccc[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP5 Q13451 1/20 0.42
CYP1A2 P05177 1/20 0.39
METAP2 P50579 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
CYP3A4 P08684 3/20 0.38
CYP3A5 P20815 2/20 0.38
XDH P47989 1/20 0.38
GRIN1 Q05586 2/20 0.36
GRIN2B Q13224 2/20 0.36
MALT1 Q9UDY8 1/20 0.36
PIK3CA P42336 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
SCN10A Q9Y5Y9 2/20 0.35
TAS2R14 Q9NYV8 2/20 0.34
SCN8A Q9UQD0 1/20 0.34
CYP2C9 P11712 1/20 0.34
SLC22A6 Q4U2R8 1/20 0.34
SLC22A8 Q8TCC7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30133235 0.80 CYP1A2 (0.49) CYP1A2METAP2CYP11B1CYP11B2CYP3A4
SCHEMBL2749165 0.80 CYP1A2 (0.49) CYP1A2METAP2CYP11B1CYP11B2CYP3A4
SCHEMBL11263619 0.76 FKBP5 (0.42) FKBP5CYP11B1CYP11B2XDHPIK3CA
SCHEMBL1477358 0.71 GRM5 (0.51) CYP11B1CYP11B2CYP3A4CYP3A5CHRNB2
SCHEMBL1476263 0.68 CHRNB2 (0.57) CYP3A4CYP3A5GRIN1GRIN2BCHRNB2
SCHEMBL1477141 0.67 GRM5 (0.50) CYP11B1CYP11B2CHRNB2CHRNA4TAS2R14
Water SCHEMBL14333714 0.67
SCHEMBL22338688 0.67 CYP1A2 (0.40) CYP1A2METAP2CYP11B1CYP11B2CYP3A4
SCHEMBL20448751 0.66 CYP11B2 (0.38) CYP1A2METAP2CYP11B1CYP11B2CYP3A4
SCHEMBL16894199 0.65 KIF11 (0.62) CYP1A2METAP2CYP11B1CYP11B2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4990512-A Insecticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-02-05 US disclosed