SCHEMBL9765990

SCHEMBL9765990

CCOC(=O)C(CCN1CCN(c2ncc(F)cn2)CC1)C(=O)c1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.54
KDM4E B2RXH2 1/20 0.52
CYP1A2 P05177 1/20 0.52
GAA P10253 1/20 0.52
CYP2C9 P11712 1/20 0.52
DRD2 P14416 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9765996 0.82 SIGMAR1 (0.52) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL9766044 0.74 SIGMAR1 (0.54) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL7246517 0.72 DRD2 (0.82) SIGMAR1KDM4ECYP1A2GAACYP2C9
Hydrochloric Acid SCHEMBL9766015 0.71 DRD2 (0.80) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL9400880 0.71 HTT (0.55) KDM4EGAA
Hydrochloric Acid SCHEMBL9766063 0.71 SIGMAR1 (0.89) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL9630285 0.70 OPRM1 (0.44) SIGMAR1KDM4ECYP2C9DRD2
SCHEMBL9765993 0.70 SIGMAR1 (1.00) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL7448827 0.70 KMT2A (0.43) KDM4ECYP1A2CYP2C9
SCHEMBL7373212 0.70 KMT2A (0.43) KDM4ECYP1A2GAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994460-A Treatment or prevention of disorders resulting from central nervous system anoxia BRISTOL-MYERS SQUIBB CO. (US) 1991-02-19 US disclosed
EP-0400661-A1 Agents for treatment of brain ischemia Bristol-Myers Squibb Company (US) 1990-12-05 EP disclosed