SCHEMBL9630285

SCHEMBL9630285

CCOC(=O)C(CCN1CCC(=C(c2ccc(F)cc2)c2ccc(F)cc2)CC1)C(C)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.44
MAPT P10636 3/20 0.44
DGKA P23743 3/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
TP53 P04637 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
ALOX15 P16050 2/20 0.44
TSHR P16473 2/20 0.44
HSD17B10 Q99714 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
HRH1 P35367 2/20 0.44
OPRK1 P41145 2/20 0.44
HIF1A Q16665 2/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
GMNN O75496 1/20 0.44
ADRB2 P07550 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9632061 0.90 OPRD1 (0.50) OPRM1MAPTDGKAALDH1A1LMNA
SCHEMBL9631391 0.87 OPRD1 (0.48) OPRM1OPRK1MEN1HTR7KMT2A
SCHEMBL9872824 0.81 HTR2A (0.56) ALDH1A1CYP2D6MEN1CYP3A4HTR2A
SCHEMBL9870722 0.78 DRD2 (0.52) OPRM1CYP2D6MEN1HTR1AADRA2A
SCHEMBL9870819 0.76 KMT2A (0.51) OPRM1ALDH1A1LMNACYP2D6MEN1
SCHEMBL10963542 0.75 HTR2A (0.54) ALDH1A1CYP2D6HRH1CYP3A4HTR2A
SCHEMBL16481505 0.75 OPRD1 (0.54) OPRM1MAPTDGKAALDH1A1LMNA
SCHEMBL9630470 0.74 MEN1 (0.45) MAPTALDH1A1LMNACYP2D6MEN1
SCHEMBL10932484 0.74 MAPT (0.49) MAPTALDH1A1LMNAHRH1HTR1A
SCHEMBL10554622 0.74 HRH3 (0.63) HRH1HTR2AKCNH2HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5079249-A Serotine antagonists at 5-HT2 level, antiallergens, antihistamines ADIR ET COMPAGNIE (FR) 1992-01-07 US disclosed
US-5071847-A BIS (ARYL) ALKENE COMPOUNDS OF HOMOPIPERIDINES USEFUL AS SEROTONIN-ANTAGONISTS ADIR ET COMPAGNIE (FR) 1991-12-10 US disclosed
US-5028607-A Antiserotonine agents ADIR ET COMPAGNIE (FR) 1991-07-02 US disclosed