SCHEMBL9767628

SCHEMBL9767628

CCCCC1Oc2ccc([N+](=O)[O-])cc2C(N)C1O

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.35
MAPT P10636 5/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MANBA O00462 1/20 0.35
ESPL1 Q14674 1/20 0.34
AKR1B1 P15121 1/20 0.34
POLB P06746 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP19A1 P11511 2/20 0.33
LMNA P02545 2/20 0.33
CACNA1C Q13936 2/20 0.33
CACNA1F O60840 1/20 0.33
CACNA1D Q01668 1/20 0.33
CACNA1S Q13698 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9767624 1.00 MAOB (0.35) MAOBMAPTNPSR1MANBAESPL1
SCHEMBL5695096 0.88 MAOB (0.38) MAOBMAPTNPSR1MANBAESPL1
SCHEMBL9767280 0.88 MANBA (0.39) MAPTNPSR1MANBAAKR1B1POLB
SCHEMBL9767276 0.88 MANBA (0.39) MAPTNPSR1MANBAAKR1B1POLB
SCHEMBL9767148 0.79 HIF1A (0.39) MAPTNPSR1AKR1B1ALDH1A1TDP1
SCHEMBL9767152 0.79 HIF1A (0.39) MAPTNPSR1AKR1B1ALDH1A1TDP1
SCHEMBL9767261 0.79 MAOB (0.36) MAOBMAPTESPL1AKR1B1POLB
SCHEMBL9766987 0.76 KCNE1 (0.41) MEN1KMT2A
SCHEMBL9767527 0.74 ESPL1 (0.42) MAPTNPSR1ESPL1AKR1B1POLB
SCHEMBL9865865 0.74 ESPL1 (0.42) MAPTNPSR1ESPL1AKR1B1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5072006-A Chemical intermeidate; hypotensive agents, muscle relaxants RECHERCHE SYNTEX FRANCE S.A. (FR) 1991-12-10 US disclosed
US-4997846-A Smooth muscle relaxants, hypotensives RESEARCHE SYNTEX FRANCE, S.A. (FR) 1991-03-05 US disclosed
EP-0377966-A2 Novel benzopyranylpyrrolinone derivatives RECHERCHE SYNTEX FRANCE SA (FR) 1990-07-18 EP disclosed