SCHEMBL9768337

SCHEMBL9768337

O=C1Cc2cc(C(O)CN3CCC(Oc4ccccn4)CC3)ccc2N1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.51
HTR1A P08908 1/20 0.49
DRD2 P14416 1/20 0.49
HTR2A P28223 1/20 0.49
GRIA1 P42261 5/20 0.42
KCNH2 Q12809 3/20 0.42
ALDH1A1 P00352 1/20 0.41
ATM Q13315 1/20 0.41
IP6K1 Q92551 1/20 0.41
KDM5A P29375 1/20 0.40
KDM1A O60341 1/20 0.39
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768289 0.86 GRIN2B (0.57) GRIN2BHTR1ADRD2HTR2AGRIA1
SCHEMBL8301786 0.75 HTR1A (0.53) GRIN2BHTR1ADRD2HTR2AKCNH2
SCHEMBL8122268 0.73 KCNH2 (0.67) GRIN2BHTR1ADRD2HTR2AKCNH2
SCHEMBL9768368 0.72 GRIN2B (0.60) GRIN2BHTR1ADRD2HTR2AKCNH2
SCHEMBL8123895 0.71 GRIN2B (0.74) GRIN2BHTR1ADRD2HTR2AKCNH2
SCHEMBL28574924 0.70 HTR2A (0.64) GRIN2BHTR1ADRD2HTR2AKCNH2
SCHEMBL8549047 0.69 GRIN1 (0.63) GRIN2BADRA1DADRA1AADRA1B
SCHEMBL15586812 0.69 KCNH2 (0.57) GRIN2BHTR1ADRD2HTR2AKCNH2
SCHEMBL10838656 0.69 GRIN2B (0.51) GRIN2BHTR1ADRD2HTR2AKCNH2
SCHEMBL29960317 0.69 GRIN2B (0.56) GRIN2BHTR1ADRD2HTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034401-A Cardiovascular disorders or antiischemia agents SYNTHELABO (FR) 1991-07-23 US disclosed