SCHEMBL9769967

SCHEMBL9769967

COC(=O)C(NC(=O)CNC(=O)OC(C)(C)C)c1cccs1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
CTSK P43235 4/20 0.42
CTSS P25774 3/20 0.42
TACR3 P29371 1/20 0.41
REN P00797 1/20 0.40
PTPRB P23467 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
CTSL P07711 1/20 0.38
SYK P43405 1/20 0.38
KLK5 Q9Y337 2/20 0.37
EPHX2 P34913 1/20 0.36
CCR2 P41597 1/20 0.35
NPFFR1 Q9GZQ6 1/20 0.35
NPFFR2 Q9Y5X5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9779450 0.89 CTSK (0.45) CYP3A4CYP2D6CYP2C9ALOX15TSHR
SCHEMBL28237555 0.81 CTSS (0.54) CTSKCTSSCTSLSYKKLK5
SCHEMBL7158579 0.79 CTSK (0.45) CYP3A4CYP2D6CYP2C9ALOX15TSHR
SCHEMBL4152673 0.78 TACR3 (0.40) CYP3A4CYP2D6CYP2C9ALOX15TSHR
SCHEMBL9769981 0.76 TACR3 (0.43) CYP3A4CYP2D6CYP2C9ALOX15TSHR
SCHEMBL9779446 0.75 CTSS (0.51) CYP3A4CYP2D6CYP2C9ALOX15TSHR
SCHEMBL3220161 0.75 CTSK (0.48) CYP3A4CYP2D6CYP2C9ALOX15TSHR
SCHEMBL3685468 0.75 CTSK (0.48) CYP3A4CYP2D6CYP2C9ALOX15TSHR
SCHEMBL11522699 0.75 CTSK (0.46) CYP3A4CYP2D6CYP2C9ALOX15TSHR
SCHEMBL1789747 0.75 CTSK (0.48) CYP3A4CYP2D6CYP2C9ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4987134-A DISORDERS OF BRAIN FUNCTIONS CASSELLA AKTIENGESELLSCHAFT (DE) 1991-01-22 US disclosed