SCHEMBL9769981

SCHEMBL9769981

COC(=O)C(NC(=O)C(N)C(=O)OC(C)(C)C)c1cccs1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 2/20 0.43
REN P00797 1/20 0.39
CTSK P43235 3/20 0.36
CTSS P25774 2/20 0.36
TSHR P16473 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALOX5 P09917 1/20 0.35
CCR2 P41597 1/20 0.34
HPGD P15428 2/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
CTSC P53634 1/20 0.33
CTSL P07711 1/20 0.33
LMNA P02545 1/20 0.33
GLA P06280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9769967 0.76 CYP3A4 (0.43) TACR3RENCTSKCTSSTSHR
SCHEMBL9779472 0.76 ALOX5 (0.43) CTSKCTSSTSHRALOX5HPGD
SCHEMBL7158579 0.76 CTSK (0.45) TACR3RENCTSKCTSSTSHR
SCHEMBL4152673 0.75 TACR3 (0.40) TACR3RENCTSKCTSSTSHR
Methane SCHEMBL11683717 0.74 TACR3 (0.50) TACR3TSHRCYP3A4CYP2D6CYP2C9
SCHEMBL7369517 0.74 REN (0.44) TACR3RENTSHRCCR2
SCHEMBL6649268 0.73 SLC1A3 (0.42) CTSKCTSSCYP2D6CYP2C9CYP2C19
SCHEMBL14217667 0.73 CTSK (0.45) RENCTSKCTSSTSHRCYP3A4
SCHEMBL5027594 0.73 CTSK (0.45) RENCTSKCTSSTSHRCYP3A4
SCHEMBL6647754 0.72 ALOX5 (0.38) CTSKCTSSALOX5HPGDCHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4987134-A DISORDERS OF BRAIN FUNCTIONS CASSELLA AKTIENGESELLSCHAFT (DE) 1991-01-22 US disclosed