SCHEMBL9770699

SCHEMBL9770699

COC(=O)c1cn2c(=O)c3cc(SC)ccc3nc2s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
MMP13 P45452 1/20 0.39
ALPG P10696 1/20 0.38
DHODH Q02127 1/20 0.35
AKR1B1 P15121 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
NPC1 O15118 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
UBE2N P61088 1/20 0.34
ICAM1 P05362 1/20 0.34
SELE P16581 1/20 0.34
VCAM1 P19320 1/20 0.34
RXFP1 Q9HBX9 2/20 0.34
TP53 P04637 1/20 0.34
KDM4E B2RXH2 2/20 0.34
POLB P06746 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPT P10636 3/20 0.33
TYMS P04818 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11014908 0.91 DHODH (0.40) MMP13ALPGDHODHAKR1B1ICAM1
SCHEMBL9770670 0.84 ALPG (0.55) ALDH1A1HPGDALPGNPC1KDM4E
SCHEMBL10696742 0.82 MMP13 (0.38) MMP13ALPGDHODHAKR1B1NPC1
SCHEMBL28345238 0.81 ALDH1A1 (0.50) ALDH1A1HPGDNPC1RXFP1TP53
SCHEMBL11397996 0.81 AKR1B1 (0.37) ALDH1A1HPGDMMP13ALPGDHODH
SCHEMBL11014615 0.76 ALPG (0.60) ALDH1A1HPGDALPGDHODHKDM4E
SCHEMBL11015093 0.71 PTAFR (0.42)
SCHEMBL11015097 0.70 MEN1 (0.39) ALDH1A1HPGDALPGL3MBTL1NPC1
SCHEMBL11018500 0.70 ALPG (0.37) ALPGAKR1B1MEN1KMT2A
SCHEMBL11270745 0.69 ALPG (0.67) ALDH1A1HPGDALPGDHODHAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5030727-A Reacting an anthronilide derivative with a thiazole derivative or a fluorozuinazolone with a neucleophile BASF AKTIENGESELLSCHAFT (DE) 1991-07-09 US disclosed
US-4282360-A ANTIALLERGENS HOFFMANN-LA ROCHE INC. (US) 1981-08-04 US disclosed
EP-0027268-A2 Quinazoline derivatives, process and intermediates for their preparation, medicaments containing them and their pharmaceutical use F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-04-22 EP disclosed