SCHEMBL9779355

SCHEMBL9779355

COC(=O)CNC(C(=O)O)c1cccs1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
TP53 P04637 3/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
THRB P10828 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TACR3 P29371 1/20 0.38
KMT2A Q03164 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALOX5 P09917 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9769954 0.87 ALOX5 (0.42) CYP2C19CYP3A4CYP2D6CYP2C9ALOX15
SCHEMBL4693687 0.86 CTSK (0.38) CYP2C19CYP3A4CYP2D6CYP2C9ALOX15
SCHEMBL9542762 0.82 L3MBTL1 (0.42) TSHRTP53POLBKMT2ANPC1
SCHEMBL9326172 0.82 ALOX5 (0.42) CYP2C19CYP3A4CYP2D6CYP2C9ALOX15
SCHEMBL6032865 0.81 CYP2C19 (0.42) CYP2C19CYP3A4CYP2D6CYP2C9ALOX15
SCHEMBL4629953 0.77 ALDH1A1 (0.54) CYP2C19CYP3A4CYP2D6CYP2C9ALOX15
SCHEMBL4152673 0.77 TACR3 (0.40) CYP2C19CYP3A4CYP2D6CYP2C9ALOX15
SCHEMBL11534783 0.76 ALOX5 (0.44) CYP2C19CYP3A4CYP2D6CYP2C9ALOX15
SCHEMBL9779583 0.75 ALDH1A1 (0.41) POLBNPSR1KMT2ANPC1SMN1; SMN2
Hydrochloric Acid SCHEMBL8845008 0.75 CYP2C19 (0.39) CYP2C19CYP3A4CYP2D6CYP2C9ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5015659-A Cognition activators to slow aging of the brain CASSELLA AKTIENGESELLSCHAFT (DE) 1991-05-14 US disclosed
EP-0388750-A1 Thienyl piperazines, process for their preparation, their use, pharmaceutical agents containing them and their production CASSELLA Aktiengesellschaft (DE) 1990-09-26 EP disclosed