SCHEMBL9784571

SCHEMBL9784571

CCc1nc(C(=O)O)c(C(=O)O)c(C)c1CC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.41
DPP4 P27487 3/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
ADORA3 P0DMS8 4/20 0.36
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
GABRA4 P48169 1/20 0.35
GABRE P78334 1/20 0.35
GABRA6 Q16445 1/20 0.35
GABRG1 Q8N1C3 1/20 0.35
GABRG3 Q99928 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31436370 0.85 HCAR2 (0.41) HCAR2DPP4DPP8DPP9ADORA3
SCHEMBL8995714 0.85 HCAR2 (0.41) HCAR2DPP4DPP8DPP9ADORA3
SCHEMBL8995696 0.85 GABRP (0.37) HCAR2DPP4DPP8DPP9ADORA3
SCHEMBL11375262 0.82 ALDH1A1 (0.40) HCAR2DPP4DPP8DPP9ADORA3
SCHEMBL29188835 0.79 GABRP (0.33) HCAR2DPP4DPP8DPP9ADORA3
SCHEMBL8995682 0.76 KMO (0.34) HCAR2DPP4DPP8DPP9ADORA3
SCHEMBL9784563 0.76 HCAR2 (0.38) HCAR2DPP4DPP8DPP9ADORA3
SCHEMBL29102125 0.73 PDE10A (0.34) HCAR2DPP4MEN1KMT2AKDM4E
SCHEMBL30968740 0.73 HCAR2 (0.33) HCAR2DPP4DPP8DPP9ADORA3
SCHEMBL21843253 0.73 NPC1 (0.48) HCAR2GABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047542-A Reaction of ketoester with unsaturated aldehyde or ketone HOECHST CELANESE CORPORATION (US) 1991-09-10 US claimed
US-4871859-A REACTING KETOESTER WITH UNSATURATED ALDEHYDE OR KETONE AND AMMONIUM SALT IN SOLVENT AND DEHYDROGENATION CATALYST HOECHST CELANESE CORPORATION 1989-10-03 US claimed
WO-1989008103-A1 PROCESS FOR PREPARING PYRIDINE CARBOXYLIC ACID ESTERS HOECHST CELANESE CORPORATION (US) 1989-09-08 WO claimed