SCHEMBL9788014

SCHEMBL9788014

O=[N+]([O-])c1sc(Nc2cccc(Br)c2)nc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.53
ADORA2A P29274 2/20 0.53
ADORA1 P30542 1/20 0.53
EGFR P00533 12/20 0.47
EPM2A O95278 1/20 0.44
PTPN1 P18031 1/20 0.44
PTPN6 P29350 1/20 0.44
PTPN9 P43378 1/20 0.44
DUSP3 P51452 1/20 0.44
PTPN11 Q06124 1/20 0.44
PTGES O14684 1/20 0.41
ALOX5 P09917 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
PKM P14618 1/20 0.41
MAPT P10636 2/20 0.40
PSMD14 O00487 1/20 0.40
LMNA P02545 1/20 0.40
PTGS2 P35354 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9788999 0.85 RAB9A (0.50) ADORA3EGFRMEN1KMT2ANPC1
SCHEMBL9788042 0.84 MAPT (0.56) ADORA3ADORA2AMEN1KMT2ANPC1
SCHEMBL9789067 0.78 LMNA (0.40) ADORA3ADORA2AADORA1MEN1KMT2A
SCHEMBL9789051 0.76 ADORA3 (0.48) ADORA3ALOX5MEN1KMT2ANPC1
SCHEMBL9789038 0.73 CA1 (0.52) ADORA3EGFRMEN1KMT2AMAPT
SCHEMBL9789114 0.72 ADORA3 (0.44) ADORA3MEN1KMT2AMAPTPSMD14
SCHEMBL9789019 0.71 KMT2A (0.44) ALOX5MEN1KMT2ANPC1MAPT
SCHEMBL6153975 0.69 ROCK2 (0.62) EGFRPTGESALOX5MEN1KMT2A
SCHEMBL8298036 0.68 PIN1 (0.72) EGFR
SCHEMBL9788026 0.68 NPC1 (0.36) ADORA3MEN1KMT2ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2078672-A None JP disclosed
US-5075326-A Fungicides, microbiocides BAYER AKTIENGESELLSCHAFT (DE) 1991-12-24 US disclosed
US-5071865-A Fungicides, bactericides BAYER AKTIENGESELLSCHAFT (DE) 1991-12-10 US disclosed
EP-0402716-A1 2-Acylamino-4-halogeno-5-nitrothiazole derivatives, process for their preparation, their use in pesticides and new intermediate products BAYER AG (DE) 1990-12-19 EP disclosed
US-4962102-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1990-10-09 US disclosed
JP-H0278672-A 4-HALOGENO-5-NITROTHIAZOLE DERIVATIVE, ITS PRODUCTION AND NOVEL INTERMEDIATE USED AS HARMFUL ORGANISM CONTROL AGENT BAYER AG 1990-03-19 JP disclosed
EP-0351662-A2 4-Halo-5-nitrothiazole derivatives, process for their preparation, their use as pesticides, and intermediates BAYER AG (DE) 1990-01-24 EP disclosed