Oxalic Acid

Oxalic Acid

SCHEMBL9788758

COc1cc2onc(CCCN3CCN(C(c4ccccc4)c4ccccc4)CC3)c2cc1OC.O=C(O)C(=O)O

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
DRD2 P14416 7/20 0.54
DRD3 P35462 7/20 0.54
DRD4 P21917 6/20 0.54
TDP1 Q9NUW8 1/20 0.46
MAPT P10636 2/20 0.46
LMNA P02545 2/20 0.46
KDM4E B2RXH2 2/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
GAA P10253 1/20 0.46
MAPK1 P28482 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9788769 0.95 DRD2 (0.58) ALDH1A1L3MBTL1DRD2DRD3DRD4
Oxalic Acid SCHEMBL9788820 0.95 ALDH1A1 (0.52) ALDH1A1L3MBTL1DRD2DRD3DRD4
SCHEMBL9879857 0.90 DRD3 (0.53) ALDH1A1L3MBTL1DRD2DRD3DRD4
SCHEMBL9788786 0.86 DRD2 (0.52) DRD2DRD3DRD4LMNA
SCHEMBL9788764 0.82 ACHE (0.46) KDM4E
Oxalic Acid SCHEMBL9788762 0.79 MEN1 (0.45) ALDH1A1DRD2DRD3DRD4TDP1
Oxalic Acid SCHEMBL9876622 0.78 HTR7 (0.48) ALDH1A1DRD2DRD3DRD4LMNA
SCHEMBL9788796 0.78 DRD2 (0.56) DRD2DRD3DRD4
SCHEMBL9788754 0.76 DRD2 (0.52) DRD2DRD3DRD4
SCHEMBL9788787 0.72 DRD2 (0.44) DRD2DRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5030639-A N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-07-09 US disclosed
US-5008264-A N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-04-16 US disclosed
US-4980365-A N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-12-25 US disclosed
EP-0299349-A2 N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-01-18 EP disclosed