Oxalic Acid

Oxalic Acid

SCHEMBL9797281

Clc1cccc(OC2CN(CC3CC3)CCc3ccccc32)c1.O=C(O)C(=O)O

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM2B Q8NHM5 10/20 0.46
SIGMAR1 Q99720 1/20 0.43
OPRK1 P41145 1/20 0.42
HRH3 Q9Y5N1 4/20 0.42
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9797472 0.94 SIGMAR1 (0.47) KDM2BSIGMAR1OPRK1HRH3THRB
Oxalic Acid SCHEMBL9797491 0.85 OPRM1 (0.48) SIGMAR1HRH3KDM4EALDH1A1TP53
SCHEMBL9797767 0.80 SIGMAR1 (0.48) SIGMAR1
SCHEMBL9797229 0.79 LMNA (0.40) SIGMAR1HRH3
SCHEMBL9797369 0.79 SIGMAR1 (0.46) KDM2BSIGMAR1HRH3
SCHEMBL9797302 0.79 GAA (0.42) SIGMAR1
SCHEMBL9797486 0.78 MEN1 (0.42) SIGMAR1TSHR
SCHEMBL9154713 0.75 SLC6A4 (0.38) SIGMAR1
SCHEMBL9797514 0.75 HRH3 (0.42) SIGMAR1OPRK1HRH3KDM4ETP53
Oxalic Acid SCHEMBL9797475 0.74 SLC6A4 (0.43) OPRK1KDM4EALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5059688-A 1-aryloxy-2,3,4,5-tetrahydro-3-benzazepine preparation HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-10-22 US disclosed
US-4988690-A Antidepressants HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-01-29 US disclosed
US-4935418-A Medical compositions of 1-aryloxy-2,3,4,5-tetrahydro-3-benzazepines and use thereof HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-19 US disclosed
US-4794181-A ANTIDEPRESSANTS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-12-27 US disclosed
EP-0096838-B1 1-ARYLOXY-2,3,4,5-TETRAHYDRO-3-BENZAZEPINES, A PROCESS FOR PREPARING THE SAME AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1987-04-01 EP disclosed
EP-0096838-A1 1-Aryloxy-2,3,4,5-tetrahydro-3-benzazepines, a process for preparing the same and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1983-12-28 EP disclosed