SCHEMBL9815960

SCHEMBL9815960

COc1ccccc1N1CCN(CC(O)COc2ccc(CC(C)=O)cc2)CC1

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.69
CACNA1G O43497 1/20 0.69
MAPT P10636 7/20 0.64
ALDH1A1 P00352 2/20 0.64
LMNA P02545 7/20 0.63
HSP90AB1 P08238 1/20 0.62
MAPK1 P28482 3/20 0.62
HTT P42858 2/20 0.62
SMN1; SMN2 Q16637 1/20 0.61
TDP1 Q9NUW8 2/20 0.61
KDM4E B2RXH2 2/20 0.61
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
HIF1A Q16665 2/20 0.61
NR1I2 O75469 1/20 0.61
NR3C1 P04150 1/20 0.61
ADRB1 P08588 1/20 0.61
HTR1A P08908 1/20 0.61
ADRA2A P08913 1/20 0.61
DRD2 P14416 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9816000 0.89 MAPT (0.64) KCNH2CACNA1GMAPTALDH1A1LMNA
SCHEMBL9815962 0.88 ABCB1 (0.77) ABCB1
SCHEMBL17313697 0.86 KCNH2 (0.78) KCNH2CACNA1GMAPTALDH1A1LMNA
SCHEMBL11817687 0.85 CACNA1G (0.80) KCNH2CACNA1GMAPTALDH1A1LMNA
SCHEMBL9815965 0.84 HTR7 (0.76) MAPTALDH1A1LMNAMAPK1MEN1
Hydrochloric Acid SCHEMBL11813716 0.84 CACNA1G (0.79) KCNH2CACNA1GMAPTALDH1A1LMNA
SCHEMBL17313690 0.81 MAPT (0.74) KCNH2CACNA1GMAPTALDH1A1LMNA
SCHEMBL9815963 0.81 ABCB1 (0.67) MEN1KMT2AABCB1
SCHEMBL9815982 0.81 KCNH2 (0.61) KCNH2CACNA1GMAPTALDH1A1LMNA
Enciprazine SCHEMBL584730 0.80 MAPT (0.74) KCNH2CACNA1GMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0167121-B1 SUBSTITUTED PHENYLPIPERAZINYL PROPANOLS, PROCESS FOR THEIR PREPARATION, THEIR USE, AND COMPOSITIONS CONTAINING THESE COMPOUNDS Beiersdorf Aktiengesellschaft (DE) 1991-10-23 EP disclosed
US-4631281-A ANTICOAGULANTS, ASTHMA, HYPOTENSIVE AGENTS, BRONCHOPILATORS, INOTROPIC AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1986-12-23 US disclosed