SCHEMBL9818889

SCHEMBL9818889

CN(C(=O)C(C#N)C(=O)c1ccc(C(F)(F)F)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.45
MLYCD O95822 3/20 0.45
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
RAPGEF3 O95398 2/20 0.41
RAPGEF4 Q8WZA2 2/20 0.41
SLC6A4 P31645 1/20 0.40
TACR1 P25103 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
NR1H3 Q13133 2/20 0.37
NR1H2 P55055 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SRD5A2 P31213 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9818892 0.94 CYP11B1 (0.43) GSK3BMLYCDCES2CES1RAPGEF3
SCHEMBL9818860 0.94 CYP11B1 (0.43) GSK3BMLYCDCES2CES1RAPGEF3
SCHEMBL9818875 0.94 MLYCD (0.43) GSK3BMLYCDCES2CES1RAPGEF3
SCHEMBL9819113 0.82 ALDH1A1 (0.42) CES2CES1RAPGEF3SMN1; SMN2ALDH1A1
SCHEMBL9819226 0.78 RAPGEF3 (0.48) RAPGEF3SMN1; SMN2TSHRLMNANPSR1
SCHEMBL1858924 0.73 GSK3B (0.56) GSK3BCES2CES1RAPGEF3RAPGEF4
SCHEMBL8309743 0.73 GSK3B (0.59) GSK3BCES2CES1RAPGEF3RAPGEF4
SCHEMBL9818928 0.72 EPHX2 (0.50) GSK3BCES2CES1RAPGEF3RAPGEF4
SCHEMBL14364710 0.72 GSK3B (0.47) GSK3BCES2CES1RAPGEF3RAPGEF4
SCHEMBL9819075 0.70 EPHX2 (0.47) GSK3BCES2CES1RAPGEF3RAPGEF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed