SCHEMBL9818892

SCHEMBL9818892

CN(C(=O)C(C#N)C(=O)c1ccc(C(F)(F)F)cc1)c1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
GPBAR1 Q8TDU6 1/20 0.43
UTS2R Q9UKP6 2/20 0.42
RAPGEF3 O95398 4/20 0.41
RAPGEF4 Q8WZA2 3/20 0.41
GSK3B P49841 1/20 0.40
MLYCD O95822 1/20 0.40
LIPE Q05469 1/20 0.40
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
LTC4S Q16873 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MGLL Q99685 1/20 0.38
KLRK1 P26718 1/20 0.37
MICA Q29983 1/20 0.37
RAET1L Q5VY80 1/20 0.37
TACR2 P21452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9818860 1.00 CYP11B1 (0.43) CYP11B1CYP11B2GPBAR1UTS2RRAPGEF3
SCHEMBL9818889 0.94 GSK3B (0.45) RAPGEF3RAPGEF4GSK3BMLYCDCES2
SCHEMBL9819113 0.90 ALDH1A1 (0.42) UTS2RRAPGEF3LIPECES2CES1
SCHEMBL9818875 0.88 MLYCD (0.43) RAPGEF3RAPGEF4GSK3BMLYCDCES2
SCHEMBL9819226 0.85 RAPGEF3 (0.48) CYP11B1CYP11B2GPBAR1RAPGEF3LIPE
SCHEMBL9818823 0.76 RHOC (0.49) RAPGEF3RAPGEF4P2RX1
SCHEMBL9819165 0.76 RHOC (0.49) RAPGEF3RAPGEF4P2RX1
SCHEMBL8201118 0.71 CHRNB2 (0.39) GPBAR1LIPEALDH1A1POLBTDP1
SCHEMBL9819360 0.70 RAPGEF3 (0.43) RAPGEF3RAPGEF4
SCHEMBL9819198 0.70 ENPP3 (0.49) RAPGEF3RAPGEF4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed