SCHEMBL9818936

SCHEMBL9818936

Cc1cc(Oc2ccc(C(F)(F)F)cc2)ccc1NC(=O)C(C#N)C(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 3/20 0.45
MAPT P10636 3/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPK1 P28482 1/20 0.40
KDR P35968 3/20 0.40
BRAF P15056 1/20 0.40
LIPE Q05469 4/20 0.39
RAPGEF3 O95398 1/20 0.39
RAPGEF4 Q8WZA2 1/20 0.39
PPARG P37231 1/20 0.38
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
S1PR2 O95136 1/20 0.37
MAPK14 Q16539 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819234 0.97 RAF1 (0.43) RAF1MAPTKDM4EMAPK1KDR
SCHEMBL9819086 0.85 RAPGEF3 (0.40) MAPTRAPGEF3RAPGEF4MEN1HTT
SCHEMBL9819360 0.85 RAPGEF3 (0.43) MAPTMAPK1RAPGEF3RAPGEF4PPARG
SCHEMBL9819062 0.83 TRPV1 (0.49) MAPTKDM4EMAPK1KDRBRAF
SCHEMBL9819084 0.82 MAPT (0.51) MAPTMAPK1MEN1HTTRAB9A
SCHEMBL9819198 0.79 ENPP3 (0.49) MAPTRAPGEF3RAPGEF4MEN1HTT
SCHEMBL9819139 0.79 TRPV1 (0.44) MAPTKDRBRAFMAPK14
SCHEMBL9819159 0.77 NPC1 (0.48) MAPTKDM4EKDRHTTRAB9A
SCHEMBL9818887 0.76 IDO1 (0.47) MAPTKDM4ERAPGEF3RAPGEF4PPARG
SCHEMBL9818928 0.76 EPHX2 (0.50) RAPGEF3RAPGEF4RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed