SCHEMBL9819360

SCHEMBL9819360

Cc1cc(Cl)ccc1NC(=O)C(C#N)C(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAPGEF3 O95398 3/20 0.43
RAPGEF4 Q8WZA2 3/20 0.43
IDO1 P14902 1/20 0.43
RAB9A P51151 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
PPARG P37231 2/20 0.41
PPARD Q03181 2/20 0.41
NR1H4 Q96RI1 2/20 0.41
GRIK1 P39086 1/20 0.40
PPARA Q07869 1/20 0.39
SLC6A3 Q01959 1/20 0.39
NPC1 O15118 1/20 0.39
CASP3 P42574 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
MAPK1 P28482 1/20 0.39
IDH1 O75874 2/20 0.39
LMNA P02545 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819116 0.90 MAPK1 (0.45) RAB9ASLC6A3NPC1CASP3SENP7
SCHEMBL9818887 0.89 IDO1 (0.47) RAPGEF3RAPGEF4IDO1RAB9ACYP1A2
SCHEMBL9819086 0.87 RAPGEF3 (0.40) RAPGEF3RAPGEF4IDO1RAB9AMEN1
SCHEMBL9819098 0.85 NPC1 (0.44) RAB9ASLC6A3NPC1CASP3SENP7
SCHEMBL9819218 0.85 NPC1 (0.43) RAB9ASLC6A3NPC1CASP3SENP7
SCHEMBL9818936 0.85 RAF1 (0.45) RAPGEF3RAPGEF4RAB9APPARGPPARD
SCHEMBL9819084 0.83 MAPT (0.51) RAB9ANPC1MAPK1LMNAMEN1
SCHEMBL9818923 0.83 MAPT (0.47) RAB9ACYP1A2CYP2D6CYP2C19NPC1
SCHEMBL9819336 0.83 RAB9A (0.49) RAB9ASLC6A3NPC1CASP3SENP7
SCHEMBL9819107 0.83 GRIK1 (0.50) RAPGEF3RAPGEF4IDO1RAB9APPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed