SCHEMBL9819218

SCHEMBL9819218

Cc1cc(Cl)ccc1NC(=O)C(C#N)C(=O)c1ccc(Br)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPT P10636 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPK1 P28482 1/20 0.41
CASP3 P42574 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
IDH1 O75874 2/20 0.41
NOX1 Q9Y5S8 1/20 0.40
SLC6A3 Q01959 1/20 0.39
DHODH Q02127 1/20 0.39
EGFR P00533 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819116 0.93 MAPK1 (0.45) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL9819098 0.88 NPC1 (0.44) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL9819336 0.88 RAB9A (0.49) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL9819360 0.85 RAPGEF3 (0.43) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL9819109 0.84 KMT2A (0.49) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL9819381 0.80 ALDH1A1 (0.48) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL9818917 0.80 ALDH1A1 (0.48) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL9819202 0.76 KMT2A (0.46) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL9818807 0.74 APP (0.52) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL9819047 0.74 ALDH1A1 (0.43) RAB9ASMN1; SMN2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034410-A Nitrile and oxo containing amides or thioamides SYNTEX (U.S.A.) INC. (US) 1991-07-23 US disclosed