SCHEMBL9819249

SCHEMBL9819249

CN1C(=O)CCN(c2ccc(C(F)(F)F)cc2)C1=O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOX4 Q9NPH5 3/20 0.46
HDAC1 Q13547 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
HSD11B1 P28845 1/20 0.45
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
PPARD Q03181 4/20 0.40
PPARA Q07869 4/20 0.40
FPR2 P25090 2/20 0.40
FPR1 P21462 1/20 0.40
LIPE Q05469 2/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CA12 O43570 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25667202 0.85 DRD2 (0.49) HSD11B1PPARDPPARAPPARG
SCHEMBL25931911 0.85 PPARD (0.48) NOX4HDAC1HSD11B1GSK3AGSK3B
SCHEMBL1261488 0.84 HSD11B1 (0.47) NOX4HDAC1CYP1A2CYP2C19HSD11B1
SCHEMBL9819261 0.84 DRD2 (0.54)
SCHEMBL20956916 0.81 RAB9A (0.54) NOX4HDAC1CYP1A2CYP2C19HSD11B1
SCHEMBL10973333 0.80 DDB1 (0.51)
SCHEMBL6418503 0.80 MEN1 (0.59) HSD11B1
SCHEMBL9819344 0.78 DRD2 (0.48) HSD11B1
Hydrochloric Acid SCHEMBL9819431 0.78 DDB1 (0.50)
SCHEMBL3824793 0.75 ALDH1A1 (0.57) NOX4FPR2FPR1LIPE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0162669-B1 ANTICONVULSIVE COMPOUNDS KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-12-11 EP disclosed
US-4588729-A Treating convulsions with dihydrouracil derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1986-05-13 US disclosed
EP-0162669-A2 Anticonvulsive compounds KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-11-27 EP disclosed