SCHEMBL9819783

SCHEMBL9819783

CCCCNC(=O)C(O[Si](C)(C)C(C)(C)C)C(N)CC1CCCCC1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.56
REN P00797 6/20 0.55
BCHE P06276 2/20 0.42
CHRNB2 P17787 5/20 0.41
CHRNB4 P30926 5/20 0.41
CHRNA3 P32297 5/20 0.41
CHRNA4 P43681 5/20 0.41
GRIN1 Q05586 2/20 0.41
GRIN2A Q12879 2/20 0.41
GRM1 Q13255 2/20 0.41
TSHR P16473 1/20 0.38
NMT2 O60551 1/20 0.38
NMT1 P30419 1/20 0.38
NAAA Q02083 1/20 0.37
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819777 1.00 METAP2 (0.56) METAP2RENBCHECHRNB2CHRNB4
SCHEMBL9819802 0.84 METAP2 (0.40) METAP2REN
SCHEMBL3564135 0.83 REN (0.48) METAP2RENBCHECHRNB2CHRNB4
SCHEMBL9819691 0.80 METAP2 (0.38) METAP2REN
SCHEMBL9819688 0.80 METAP2 (0.38) METAP2REN
SCHEMBL3565758 0.74 REN (0.39) METAP2RENBCHECHRNB2CHRNB4
SCHEMBL3565755 0.74 REN (0.39) METAP2RENBCHECHRNB2CHRNB4
SCHEMBL7724633 0.72 USP2 (0.39)
SCHEMBL7355197 0.72 METAP2 (1.00) METAP2RENCHRNB2CHRNB4CHRNA3
SCHEMBL9684341 0.71 REN (1.00) METAP2RENBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034376-A Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1991-07-23 US disclosed
US-4935405-A Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1990-06-19 US disclosed
US-4814342-A Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1989-03-21 US disclosed
EP-0266950-A2 Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1988-05-11 EP disclosed