SCHEMBL9819802

SCHEMBL9819802

CNC(=O)[C@H](O[Si](C)(C)C(C)(C)C)[C@@H](N)CC1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 10/20 0.40
METAP1 P53582 5/20 0.40
REN P00797 2/20 0.37
CTSK P43235 2/20 0.35
CTSS P25774 1/20 0.35
MMP1 P03956 1/20 0.34
MMP3 P08254 1/20 0.34
AAK1 Q2M2I8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819691 0.86 METAP2 (0.38) METAP2METAP1RENCTSKCTSS
SCHEMBL9819688 0.86 METAP2 (0.38) METAP2METAP1RENCTSKCTSS
SCHEMBL9819777 0.84 METAP2 (0.56) METAP2REN
SCHEMBL9819783 0.84 METAP2 (0.56) METAP2REN
SCHEMBL7441667 0.83 REN (0.38) METAP2METAP1RENCTSKCTSS
SCHEMBL3564135 0.73 REN (0.48) METAP2RENCTSK
SCHEMBL9514512 0.72 METAP2 (0.62) METAP2METAP1REN
SCHEMBL9514503 0.72 METAP2 (0.62) METAP2METAP1REN
SCHEMBL9514498 0.72 METAP2 (0.62) METAP2METAP1REN
SCHEMBL7268415 0.72 CTSK (0.37) METAP2RENCTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5034376-A Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1991-07-23 US disclosed
US-4935405-A Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1990-06-19 US disclosed
US-4814342-A Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1989-03-21 US disclosed
EP-0266950-A2 Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1988-05-11 EP disclosed