SCHEMBL9822735

SCHEMBL9822735

CNS(=O)(=O)c1cc2c(c(C(=O)Cl)c1)OC(C)C2

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.44
BRD4 O60885 1/20 0.35
PNMT P11086 1/20 0.35
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867437 0.88 PARP1 (0.45) PARP1BRD4TDP1
SCHEMBL9868222 0.76 ALDH1A1 (0.40) PARP1BRD4PNMT
SCHEMBL9868217 0.76 BRD4 (0.37) PARP1BRD4PNMTTDP1
SCHEMBL10810657 0.75 PARP1 (0.42) PARP1PNMT
SCHEMBL10805978 0.75 POLR1A (0.37) PARP1BRD4
SCHEMBL9867744 0.75 PARP1 (0.47) PARP1BRD4TDP1
SCHEMBL10815005 0.73 PARP1 (0.33) PARP1
SCHEMBL10814991 0.73 BRD4 (0.48) PARP1BRD4TDP1
Hydrochloric Acid SCHEMBL10810407 0.73 DRD2 (0.50)
SCHEMBL11116671 0.72 PARP1 (0.32) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231139-B1 DIHYDROBENZOFURANE AND CHROMANE CARBOXAMIDE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS NEUROLEPTICS Laboratoires DELAGRANGE (FR) 1991-12-04 EP claimed
US-5006570-A Dihydrobenzofuran- and chroman-carboxamide derivatives, processes for the preparation thereof and use thereof as neuroleptics LABORATOIRES DELAGRANGE (FR) 1991-04-09 US disclosed