SCHEMBL9822980

SCHEMBL9822980

O=C1C2CC(C(=O)N1CCCCN1CCN(c3ccc4ccccc4n3)CC1)C1C2C2C3CC4C2C4C31

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.67
HTR3A P46098 8/20 0.52
HTR7 P34969 1/20 0.52
HRH1 P35367 1/20 0.52
SLC6A4 P31645 1/20 0.49
HRH3 Q9Y5N1 1/20 0.48
DRD2 P14416 1/20 0.48
DRD3 P35462 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9600934 0.83 HTR1A (0.69) HTR1AHTR3AHTR7HRH1HRH3
SCHEMBL3676077 0.78 HTR1A (0.95) HTR1AHTR3AHTR7SLC6A4HRH3
SCHEMBL9539310 0.77 DRD2 (0.64) HTR1ADRD2
SCHEMBL9822816 0.77
SCHEMBL10556971 0.76 HTR1A (0.55) HTR1AHRH3
SCHEMBL10465797 0.75 HTR1A (0.76) HTR1AHTR7SLC6A4DRD2DRD3
SCHEMBL9822899 0.74 DRD2 (0.67) HTR1AHTR7DRD2DRD3
SCHEMBL9602546 0.74 HTR1A (0.67) HTR1AHTR3AHTR7HRH1HRH3
SCHEMBL10555981 0.74 HTR1A (0.48) HTR1AHTR3AHTR7HRH1DRD2
SCHEMBL3679755 0.72 HTR1A (0.65) HTR1AHTR3AHTR7HRH1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4797488-A N-((4-(PHENYL OR HETEROCYCLIC)PIPERAZIN-1-YL)ALKYL)-1,5-METHANOCYCLOPENT(D)AZEPINE-2,4 -DIONES; ANXIOLYTIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1989-01-10 US claimed
WO-1988007529-A1 PSYCHOTROPIC POLYCYCLIC IMIDES AMERICAN HOME PRODUCTS CORPORATION (US) 1988-10-06 WO claimed
EP-0286263-B1 PSYCHOTROPIC POLYCYCLIC IMIDES AMERICAN HOME PRODUCTS CORPORATION (US) 1991-05-15 EP disclosed