SCHEMBL9824013

SCHEMBL9824013

COc1ccc(Cl)cc1C(=C(c1ccccc1)c1ccccc1)n1ccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.46
ADRB1 P08588 3/20 0.46
ADRB3 P13945 3/20 0.46
TSHR P16473 2/20 0.42
KCNMA1 Q12791 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2C19 P33261 2/20 0.40
ALDH1A1 P00352 2/20 0.40
NR1I2 O75469 1/20 0.40
NR3C1 P04150 1/20 0.40
HTR1A P08908 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CNR1 P21554 1/20 0.40
TBXA2R P21731 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
SLC6A4 P31645 1/20 0.40
ADRA1A P35348 1/20 0.40
OPRK1 P41145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823697 0.88 ADRB2 (0.48) ADRB2ADRB1ADRB3NR1I2NR3C1
SCHEMBL9823712 0.83 IDO1 (0.45) ADRB2ADRB1ADRB3KCNMA1NR1I2
SCHEMBL9823802 0.79 KMT2A (0.44) TSHRKCNMA1CYP1A2CYP2C19ALDH1A1
SCHEMBL4286867 0.78 KCNMA1 (0.52) ADRB2ADRB1ADRB3TSHRKCNMA1
SCHEMBL9824008 0.70 CYP19A1 (0.41) ADRB2ADRB1ADRB3KCNMA1ALDH1A1
SCHEMBL9823745 0.70 CYP19A1 (0.41) ADRB2ADRB1ADRB3KCNMA1ALDH1A1
SCHEMBL10504932 0.70 CYP19A1 (0.44) ADRB2ADRB1ADRB3TSHRCYP1A2
SCHEMBL10504929 0.70 CYP19A1 (0.44) ADRB2ADRB1ADRB3TSHRCYP1A2
SCHEMBL6103175 0.69 POLB (0.66) TSHRCYP1A2CYP2C19ALDH1A1KDM4E
SCHEMBL9823586 0.68 SMN1; SMN2 (0.40) ALDH1A1MAPK1MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227100-B1 N-VINYLIMIDAZOLES AND -TRIAZOLES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1991-04-03 EP claimed
EP-0227100-B1 N-VINYLIMIDAZOLES AND -TRIAZOLES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1991-04-03 EP disclosed