SCHEMBL9825435

SCHEMBL9825435

COC(=O)OC1=CCCN(CC2COc3ccccc3C2)C1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.47
HTR1A P08908 1/20 0.46
OPRM1 P35372 1/20 0.44
OPRL1 P41146 1/20 0.44
KCNH2 Q12809 1/20 0.44
MALT1 Q9UDY8 1/20 0.41
LMNA P02545 1/20 0.38
MTNR1A P48039 2/20 0.38
FEN1 P39748 1/20 0.38
DRD2 P14416 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HDAC1 Q13547 1/20 0.37
TP53 P04637 2/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9825052 0.99 SIGMAR1 (0.47) SIGMAR1HTR1AOPRM1OPRL1KCNH2
SCHEMBL9824923 0.90 MALT1 (0.42) SIGMAR1HTR1AOPRM1OPRL1KCNH2
Hydrochloric Acid SCHEMBL9824811 0.89 MALT1 (0.41) SIGMAR1HTR1AOPRM1OPRL1KCNH2
SCHEMBL9692793 0.84 SIGMAR1 (0.49) SIGMAR1HTR1AOPRM1OPRL1KCNH2
Hydrochloric Acid SCHEMBL9692845 0.83 SIGMAR1 (0.48) SIGMAR1HTR1AOPRM1OPRL1KCNH2
SCHEMBL9824725 0.82 DRD2 (0.53) MTNR1ADRD2
SCHEMBL9825168 0.81 SIGMAR1 (0.47) SIGMAR1HTR1AOPRM1OPRL1KCNH2
Hydrochloric Acid SCHEMBL9825725 0.81 DRD2 (0.53) MTNR1ADRD2
Hydrochloric Acid SCHEMBL9824633 0.80 SIGMAR1 (0.46) SIGMAR1HTR1AOPRM1OPRL1KCNH2
SCHEMBL9824689 0.76 MTNR1A (0.46) MTNR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0252005-B1 HYDROGENATED 1-BENZOOXACYCLOALKYL-PYRIDINE CARBOXYLIC-ACID COMPOUNDS CIBA-GEIGY AG (CH) 1991-07-10 EP claimed
EP-0252005-A1 Hydrogenated 1-benzooxacycloalkyl-pyridine carboxylic-acid compounds CIBA-GEIGY AG (CH) 1988-01-07 EP claimed
EP-0252005-B1 HYDROGENATED 1-BENZOOXACYCLOALKYL-PYRIDINE CARBOXYLIC-ACID COMPOUNDS CIBA-GEIGY AG (CH) 1991-07-10 EP disclosed
EP-0252005-A1 Hydrogenated 1-benzooxacycloalkyl-pyridine carboxylic-acid compounds CIBA-GEIGY AG (CH) 1988-01-07 EP disclosed