SCHEMBL9824725

SCHEMBL9824725

COC(=O)OC1=CCCN(CC2COc3ccccc3O2)C1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.53
ADRA2A P08913 2/20 0.51
ADRA2B P18089 2/20 0.51
ADRA2C P18825 2/20 0.51
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
SCN1A P35498 1/20 0.49
SCN2A Q99250 1/20 0.49
SCN3A Q9NY46 1/20 0.49
MTNR1A P48039 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9825725 0.99 DRD2 (0.53) DRD2ADRA2AADRA2BADRA2CADRA1D
SCHEMBL9824689 0.90 MTNR1A (0.46) DRD2ADRA2AADRA2BADRA2CADRA1D
SCHEMBL567418 0.84 DRD2 (0.53) DRD2ADRA2AADRA2BADRA2CADRA1D
Hydrochloric Acid SCHEMBL9690277 0.83 DRD2 (0.53) DRD2ADRA2AADRA2BADRA2CADRA1D
SCHEMBL9825435 0.82 SIGMAR1 (0.47) DRD2MTNR1A
SCHEMBL9825208 0.81 DRD2 (0.53) DRD2ADRA2AADRA2BADRA2CADRA1D
Hydrochloric Acid SCHEMBL9825052 0.81 SIGMAR1 (0.47) DRD2MTNR1A
Hydrochloric Acid SCHEMBL9825333 0.80 DRD2 (0.53) DRD2ADRA2AADRA2BADRA2CADRA1D
SCHEMBL567307 0.77 ADRA2A (0.60) DRD2ADRA2AADRA2BADRA2CADRA1D
SCHEMBL9824923 0.76 MALT1 (0.42) DRD2MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0252005-B1 HYDROGENATED 1-BENZOOXACYCLOALKYL-PYRIDINE CARBOXYLIC-ACID COMPOUNDS CIBA-GEIGY AG (CH) 1991-07-10 EP claimed
EP-0252005-A1 Hydrogenated 1-benzooxacycloalkyl-pyridine carboxylic-acid compounds CIBA-GEIGY AG (CH) 1988-01-07 EP claimed
EP-0252005-B1 HYDROGENATED 1-BENZOOXACYCLOALKYL-PYRIDINE CARBOXYLIC-ACID COMPOUNDS CIBA-GEIGY AG (CH) 1991-07-10 EP disclosed
EP-0252005-A1 Hydrogenated 1-benzooxacycloalkyl-pyridine carboxylic-acid compounds CIBA-GEIGY AG (CH) 1988-01-07 EP disclosed