SCHEMBL9825753

SCHEMBL9825753

CCSC1=NOC(CNC(=O)CN(Cc2cccc3ccccc23)C(=O)OCc2ccccc2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FNTA P49354 2/20 0.36
FNTB P49356 2/20 0.36
TGM2 P21980 5/20 0.36
FSHR P23945 1/20 0.35
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CASP1 P29466 2/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ITGB3 P05106 1/20 0.32
ITGAV P06756 1/20 0.32
ITGA2B P08514 1/20 0.32
TNKS O95271 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4938340 0.88 TGM2 (0.47) TGM2ALDH1A1CASP1HDAC1HDAC6
SCHEMBL9825626 0.87 TGM2 (0.37) FNTAFNTBTGM2FSHRALDH1A1
SCHEMBL9825413 0.87 TGM2 (0.37) FNTAFNTBTGM2FSHRALDH1A1
SCHEMBL9825407 0.78 TGM2 (0.42) TGM2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL9826249 0.77 ALDH1A1 (0.46) TGM2ALDH1A1CYP1A2CYP3A4ITGB3
SCHEMBL10795296 0.74 TGM2 (0.44) TGM2ALDH1A1CYP1A2HSD17B10ITGB3
SCHEMBL9825150 0.73 KMT2A (0.43) FNTAFNTBALDH1A1CASP1HDAC1
SCHEMBL9825819 0.72 TDP1 (0.47) CYP1A2CYP2C19CASP1HDAC1HDAC6
SCHEMBL9826660 0.72 TGM2 (0.49) TGM2ITGB3ITGAVITGA2B
SCHEMBL9825257 0.71 TGM2 (0.61) TGM2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237082-B1 3,5-DISUBSTITUTED 4,5-DIHYDROISOXAZOLES AS TRANSGLUTAMINASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1991-05-29 EP disclosed
US-4929630-A SKIN DISORDERS, ACNE, 4,5-DIHYDROISOOXAZOLE PEPTIDES SYNTEX (U.S.A.) INC. (US) 1990-05-29 US disclosed
US-4912120-A Containing amine and amide substitution SYNTEX (U.S.A.) INC. (US) 1990-03-27 US disclosed
EP-0237082-A2 3,5-disubstituted 4,5-dihydroisoxazoles as transglutaminase inhibitors SYNTEX (U.S.A.) INC. (US) 1987-09-16 EP disclosed