SCHEMBL9826050

SCHEMBL9826050

C1=C(c2ccccc2)CCN(CCCOc2cccc3cnccc23)C1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 1/20 0.55
SIGMAR1 Q99720 2/20 0.54
PARP1 P09874 5/20 0.49
DRD3 P35462 4/20 0.47
DRD2 P14416 3/20 0.47
DRD4 P21917 3/20 0.47
HRH3 Q9Y5N1 1/20 0.47
HTR1A P08908 1/20 0.45
SLC6A4 P31645 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9826723 0.99 KCNA3 (0.54) KCNA3SIGMAR1PARP1DRD3DRD2
SCHEMBL9825804 0.79 SIGMAR1 (0.53) SIGMAR1PARP1DRD3DRD2DRD4
SCHEMBL9825581 0.78 HRH3 (0.76) KCNA3SIGMAR1DRD3DRD2HRH3
SCHEMBL9825701 0.77 HTR1A (0.70) DRD3DRD2DRD4HTR1ASLC6A4
SCHEMBL9825914 0.75 HRH3 (0.57) KCNA3DRD3DRD2HRH3HTR1A
SCHEMBL9825650 0.74 DRD3 (0.57) KCNA3DRD3DRD2HRH3HTR1A
Hydrochloric Acid SCHEMBL9825840 0.74 DRD3 (0.56) KCNA3DRD3DRD2HRH3HTR1A
SCHEMBL9825205 0.74 HTR1A (0.68) DRD3DRD2DRD4HTR1ASLC6A4
SCHEMBL9473840 0.71 SIGMAR1 (0.92) SIGMAR1PARP1DRD3DRD2DRD4
SCHEMBL9467947 0.71 SIGMAR1 (0.66) SIGMAR1PARP1DRD3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237781-B1 PHENYL AND HETEROCYCLIC TETRAHYDROPYRIDYL AND PIPERAZINYL ALKOXY-BENZHETEROCYCLIC COMPOUNDS AS ANTIPSYCHOTIC AGENTS WARNER-LAMBERT COMPANY (US) 1991-04-24 EP claimed
US-4704390-A SCHIZOPHRENIA WARNER-LAMBERT COMPANY (US) 1987-11-03 US claimed
EP-0237781-A2 Phenyl and heterocyclic tetrahydropyridyl and piperazinyl alkoxy-benzheterocyclic compounds as antipsychotic agents WARNER-LAMBERT COMPANY (US) 1987-09-23 EP claimed
EP-0237781-B1 PHENYL AND HETEROCYCLIC TETRAHYDROPYRIDYL AND PIPERAZINYL ALKOXY-BENZHETEROCYCLIC COMPOUNDS AS ANTIPSYCHOTIC AGENTS WARNER-LAMBERT COMPANY (US) 1991-04-24 EP disclosed
US-4803203-A SCHIZOPHRENIA, NEUOLEPTIC AGENTS WARNER-LAMBERT COMPANY (US) 1989-02-07 US disclosed
US-4704390-A SCHIZOPHRENIA WARNER-LAMBERT COMPANY (US) 1987-11-03 US disclosed
EP-0237781-A2 Phenyl and heterocyclic tetrahydropyridyl and piperazinyl alkoxy-benzheterocyclic compounds as antipsychotic agents WARNER-LAMBERT COMPANY (US) 1987-09-23 EP disclosed