SCHEMBL9826458

SCHEMBL9826458

CCCCNc1cc2ccccc2o1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.52
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
MAOB P27338 3/20 0.46
MAOA P21397 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.44
TLR8 Q9NR97 1/20 0.44
CYP2D6 P10635 1/20 0.42
HIF1A Q16665 1/20 0.42
TAS1R3 Q7RTX0 1/20 0.42
TAS1R1 Q7RTX1 1/20 0.42
ELANE P08246 1/20 0.41
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
STAT1 P42224 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424398 0.95 HDAC3 (0.48) HDAC3CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9826049 0.90 MAOB (0.51) HDAC3MAOBMAOACYP2D6HIF1A
SCHEMBL140394 0.82 NPC1 (0.51) HDAC3MAOBMAOACYP2D6HIF1A
Hydrochloric Acid SCHEMBL9826526 0.81 NPC1 (0.50) HDAC3MAOBMAOACYP2D6HIF1A
SCHEMBL19187891 0.80 CA12 (0.41) HDAC3MAOANPC1RAB9AALDH1A1
SCHEMBL5383838 0.79 LOXL2 (0.42) MAOBMAOAL3MBTL1CYP2D6HIF1A
SCHEMBL8158782 0.79 RECQL (0.46) MAOBL3MBTL1CYP2D6HIF1ATAS1R3
SCHEMBL9132475 0.76 NPC1 (0.56) HDAC3CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8947868 0.74 ALDH1A1 (0.50) MAOBL3MBTL1TAS1R3TAS1R1NPC1
SCHEMBL10169817 0.74 RIPK1 (0.50) HDAC3MAOBMAOAL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0283522-B1 TRIAZINE DERIVATIVE, PRODUCTION THEREOF, AND HERBICIDE CONTAINING SAME AS EFFECTIVE INGREDIENT IDEMITSU KOSAN COMPANY LIMITED (JP) 1991-02-27 EP disclosed
US-4932998-A LOW PHYTOTOXICITY FOR PADDY RICE PLANTS IDEMITSU KOSAN COMPANY LIMITED (JP) 1990-06-12 US disclosed
EP-0283522-A1 TRIAZINE DERIVATIVE, PRODUCTION THEREOF, AND HERBICIDE CONTAINING SAME AS EFFECTIVE INGREDIENT IDEMITSU KOSAN COMPANY LIMITED (JP) 1988-09-28 EP disclosed