SCHEMBL9826846

SCHEMBL9826846

CCOC(=O)COc1ccc(C(C)CN2CCOC(c3csc(C(F)(F)F)n3)C2)cc1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.34
POLB P06746 1/20 0.33
TBXAS1 P24557 1/20 0.33
ACACB O00763 1/20 0.33
ALDH1A1 P00352 4/20 0.33
MAPT P10636 2/20 0.33
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
KDM4E B2RXH2 3/20 0.32
HSD17B10 Q99714 2/20 0.32
TP53 P04637 1/20 0.32
HPGD P15428 1/20 0.32
NPSR1 Q6W5P4 2/20 0.32
GAA P10253 2/20 0.32
HIF1A Q16665 1/20 0.32
ALOX15 P16050 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
METAP1 P53582 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9825542 0.92 SMN1; SMN2 (0.37) SMN1; SMN2ACACBALDH1A1HPGD
SCHEMBL9825575 0.91 ALDH1A1 (0.39) SMN1; SMN2ALDH1A1KDM4EGRIN1GRIN2B
SCHEMBL9825436 0.90 PIK3CA (0.35) SMN1; SMN2ACACBALDH1A1GRIN1GRIN2B
SCHEMBL9825803 0.88 MCHR1 (0.34) SMN1; SMN2ALDH1A1TP53GRIN2B
SCHEMBL9825905 0.86 ALDH1A1 (0.38) ALDH1A1KDM4E
SCHEMBL9827149 0.86 ALDH1A1 (0.37) ALDH1A1KDM4EGRIN1GRIN2B
SCHEMBL9826520 0.84 CNR2 (0.34) KDM4E
SCHEMBL9825690 0.84 ALDH1A1 (0.39) ACACBALDH1A1KDM4E
SCHEMBL9827456 0.83 ALDH1A1 (0.39) ALDH1A1KDM4ETP53GAA
SCHEMBL8880116 0.83 ADRB2 (0.36) POLBTBXAS1ALDH1A1MAPTADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0239815-B1 SUBSTITUTED THIAZOLES AND OXAZOLES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1991-07-24 EP disclosed