SCHEMBL9828660

SCHEMBL9828660

COc1cc2c(cc1OC)CC(O)(CC(=O)O)CC2

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.39
NPSR1 Q6W5P4 2/20 0.39
NPC1 O15118 1/20 0.38
KMT2A Q03164 1/20 0.38
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37
SLC6A4 P31645 1/20 0.37
PKM P14618 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 2/20 0.36
TSHR P16473 1/20 0.36
ACHE P22303 1/20 0.35
ALOX15 P16050 1/20 0.35
THRB P10828 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
AKR1B1 P15121 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10793715 0.79 PKM (0.38) HSD17B10NPSR1MAOAMAOBSLC6A4
SCHEMBL9828092 0.77 RBP1 (0.40) HSD17B10ALDH1A1KDM4ETSHR
SCHEMBL6817239 0.73 ALDH1A1 (0.42) HSD17B10KMT2AALDH1A1KDM4ETSHR
SCHEMBL10794322 0.70 SLC18A2 (0.41) PKM
SCHEMBL8669417 0.69 DGAT1 (0.52) KMT2AALDH1A1KDM4E
SCHEMBL11561345 0.69 CYP3A4 (0.46) HSD17B10NPSR1PKMALDH1A1TSHR
SCHEMBL28071031 0.68 CYP3A4 (0.38) HSD17B10KMT2AALDH1A1KDM4ETSHR
SCHEMBL11674029 0.68 HTT (0.42) HSD17B10NPSR1KMT2AALDH1A1KDM4E
SCHEMBL7828042 0.68 KDM4E (0.41) KMT2AMAOBALDH1A1KDM4ECYP3A4
SCHEMBL7289365 0.68 L3MBTL4 (0.38) KMT2AMAOAMAOBSLC6A4PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0177960-B1 DERIVATIVES OF TETRAHYDRONAPHTHALENE, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM HOFFMANN LA ROCHE (CH) 1991-03-20 EP disclosed
US-4680310-A HYPOTENSIVE AGENTS HOFFMANN-LA ROCHE INC. (US) 1987-07-14 US disclosed
EP-0177960-A2 Derivatives of tetrahydronaphthalene, process and intermediates for their preparation and medicines containing them F. HOFFMANN-LA ROCHE AG (CH) 1986-04-16 EP disclosed