SCHEMBL9829142

SCHEMBL9829142

Cc1ccc(-c2csc(C(=O)O)n2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.55
KDM4E B2RXH2 7/20 0.55
POLB P06746 2/20 0.55
GAA P10253 2/20 0.55
HTT P42858 2/20 0.55
ALDH1A1 P00352 6/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
MAPT P10636 7/20 0.55
SMN1; SMN2 Q16637 5/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
SREBF2 Q12772 1/20 0.54
NPC1 O15118 5/20 0.52
TDP1 Q9NUW8 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
GSTO1 P78417 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6658975 0.85 RAB9A (0.61) RAB9AKDM4EPOLBGAAHTT
SCHEMBL4413970 0.84 KDM4E (0.70) RAB9AKDM4EPOLBGAAHTT
SCHEMBL167820 0.84 RAB9A (0.58) RAB9AKDM4EPOLBGAAHTT
SCHEMBL27604873 0.83 KDM4E (0.58) RAB9AKDM4EPOLBGAAHTT
SCHEMBL3934931 0.83 ALDH1A1 (0.56) RAB9AKDM4EGAAHTTALDH1A1
SCHEMBL24136180 0.83 KDM4E (0.50) RAB9AKDM4EPOLBGAAHTT
SCHEMBL3613493 0.83 RAB9A (0.63) RAB9AKDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL31401011 0.83 LMNA (0.55) RAB9AKDM4EPOLBGAAHTT
SCHEMBL5734275 0.82 KDM4E (0.51) RAB9AKDM4EPOLBGAAHTT
SCHEMBL9613335 0.82 RAB9A (0.54) RAB9AKDM4EPOLBGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119192103-A Five-membered heterocyclic amide compound, preparation method and application thereof, and bactericide 贵州大学 2024-12-27 CN disclosed
US-20220175775-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS PGE2 RECEPTOR MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2022-06-09 US disclosed
US-11241431-B2 N-substituted indole derivatives as PGE2 receptor modulators IDORSIA PHARMACEUTICALS LTD (CH) 2022-02-08 US disclosed
US-20200289507-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS PGE2 RECEPTOR MODULATORS IDORSIA PHARMACEUTICALS LTD (CH) 2020-09-17 US disclosed
US-9828351-B2 Enzyme interacting agents MONASH UNIVERSITY (AU) 2017-11-28 US disclosed
US-20170190698-A1 ENZYME INTERACTING AGENTS CENTRAL ADELAIDE LOCAL HEALTH NETWORK INCORPORATED (AU) 2017-07-06 US disclosed
US-7893084-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM CANADA LTD. (CA) 2011-02-22 US disclosed
US-7576079-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2009-08-18 US disclosed
US-20090087409-A1 Viral Polymerase Inhibitors BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2009-04-02 US disclosed
EP-1891951-A1 Viral polymerase inhibitors BOEHRINGER INGELHEIM (CANADA) LTD. (CA) 2008-02-27 EP disclosed
US-7332614-B2 Process for cross coupling indoles BOEHRINGER INGELHEIM INTERNATIONAL, GMBH (DE) 2008-02-19 US disclosed
EP-0321115-B1 CARBOXAMIDE DERIVATIVES HAVING TETRAZOLE AND THIAZOLE RINGS AND THEIR USE SAWAI PHARMACEUTICAL CO., LTD. (JP) 1991-08-14 EP disclosed
US-4946855-A ANTIALLERGIC SAWAI PHARMACEUTICAL CO., LTD. (JP) 1990-08-07 US disclosed
EP-0321115-A1 Carboxamide derivatives having tetrazole and thiazole rings and their use SAWAI PHARMACEUTICAL CO., LTD. (JP) 1989-06-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090087409-A1 Viral Polymerase Inhibitors NR2C2, NR4A1, MED25 RAB9A 3802/4885KDM4E 3438/4885POLB 166/4885
US-20200289507-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS PGE2 RECEPTOR MODULATORS PTGER1, PTGER4, PTGER2 RAB9A 3072/4885KDM4E 2755/4885POLB 3255/4885
US-20220175775-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS PGE2 RECEPTOR MODULATORS PTGER1, PTGER4, PTGER2 RAB9A 3072/4885KDM4E 2755/4885POLB 3255/4885
US-20170190698-A1 ENZYME INTERACTING AGENTS SMPD1, SMPD2, ASAH1 RAB9A 3204/4885KDM4E 3234/4885POLB 851/4885
US-11241431-B2 N-substituted indole derivatives as PGE2 receptor modulators PTGER1, PTGER4, PTGER2 RAB9A 3072/4885KDM4E 2755/4885POLB 3255/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.