SCHEMBL9830748

SCHEMBL9830748

COC(=O)C1C(=O)Nc2cc(N)c(N)cc21

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
KDM4E B2RXH2 5/20 0.34
MAPT P10636 7/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TDP2 O95551 1/20 0.34
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
HSD17B10 Q99714 2/20 0.32
ALOX15 P16050 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
KMT2A Q03164 1/20 0.32
ITGA4 P13612 1/20 0.32
USP2 O75604 1/20 0.32
GAA P10253 1/20 0.32
NLRP3 Q96P20 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833771 0.84 MAPT (0.38) ALDH1A1KDM4EMAPTRAB9AHSD17B10
SCHEMBL9830583 0.84 MAPT (0.38) ALDH1A1KDM4EMAPTRAB9AHSD17B10
SCHEMBL9832663 0.84 TDP2 (0.51) ALDH1A1KDM4EMAPTL3MBTL1TDP2
SCHEMBL9832401 0.82 MAPT (0.33) ALDH1A1KDM4EMAPTL3MBTL1NPC1
SCHEMBL9834567 0.80 ALDH1A1 (0.35) ALDH1A1KDM4EMAPTL3MBTL1TDP2
SCHEMBL4270503 0.76 TP53 (0.45) ALDH1A1KDM4EMAPTKMT2A
SCHEMBL4850477 0.76 MAPT (0.44) ALDH1A1KDM4EMAPTL3MBTL1KMT2A
SCHEMBL15075740 0.76 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTHSD17B10KMT2A
SCHEMBL9833467 0.76 CDYL2 (0.48) KMT2A
SCHEMBL7681777 0.74 MAPT (0.58) ALDH1A1KDM4EMAPTL3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed
CN-85103724-B Process for preparing pyrrolobenzimidazoles 曼海姆伯灵格股份公司 1988-07-06 CN disclosed
CN-85103724-A The method for preparing novel pyrrolo-benzoglyoxaline 1986-07-02 CN disclosed