SCHEMBL9830883

SCHEMBL9830883

Nc1n[nH]cc1C(=O)c1ccncc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
LTA4H P09960 1/20 0.42
LMNA P02545 1/20 0.42
PDE3B Q13370 2/20 0.40
PDE3A Q14432 2/20 0.40
NAPRT Q6XQN6 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MPO P05164 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
ALDH1A1 P00352 1/20 0.37
CHRM4 P08173 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3982930 0.84 MAPT (0.52) KMT2AMEN1LMNAHSD17B10ALDH1A1
SCHEMBL9832213 0.81 LTA4H (0.44) KMT2AMEN1LTA4HALDH1A1CCNA2
SCHEMBL7369952 0.81 ALDH1A1 (0.48) LMNAL3MBTL1ALDH1A1CDK2
SCHEMBL9832465 0.81 KMT2A (0.49) KMT2AMEN1
SCHEMBL7399203 0.79 NPC1 (0.54) KMT2AMEN1LMNANPSR1ALDH1A1
SCHEMBL5821548 0.76 PTPN1 (0.35) KMT2AMEN1KDM4ECYP1A2CYP3A4
SCHEMBL9832118 0.73 POLB (0.51) KMT2ANPSR1ALDH1A1CDK2
SCHEMBL9831962 0.73 PARP1 (0.47) KMT2AMEN1ALDH1A1CCNA2CDK2
SCHEMBL5793588 0.72 KMT2A (0.49) KMT2ALMNANAPRTKDM4EL3MBTL1
SCHEMBL523863 0.72 MAPT (0.49) KMT2AMEN1LMNANPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129846-B1 (3-AMINO-1H-PYRAZOL-4-YL)(ARYL)METHANONES AMERICAN CYANAMID COMPANY (US) 1991-05-08 EP claimed
US-4980472-A REACTING ACETONITRILE DERIVATIVE WITH AMINOGUANIDINE DERIVATIVE AMERICAN CYANAMID COMPANY (US) 1990-12-25 US claimed
US-4900836-A (3-amino-1H-pyrazol-4-yl) (aryl)methanones AMERICAN CYANAMID COMPANY (US) 1990-02-13 US claimed
EP-0129846-A2 (3-Amino-1H-pyrazol-4-yl)(aryl)methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP claimed