SCHEMBL7399203

SCHEMBL7399203

COc1ccc(C(=O)c2c[nH]nc2N)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
NPSR1 Q6W5P4 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 2/20 0.50
TP53 P04637 1/20 0.50
KMT2A Q03164 3/20 0.49
MAPT P10636 4/20 0.48
HTT P42858 2/20 0.48
GAA P10253 2/20 0.48
MEN1 O00255 2/20 0.47
LMNA P02545 1/20 0.47
MAPK1 P28482 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
HPGD P15428 1/20 0.47
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
PARP1 P09874 1/20 0.47
PARP10 Q53GL7 1/20 0.47
PARP2 Q9UGN5 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831105 0.84 TUBB1 (0.49) NPC1RAB9ANPSR1KMT2AMAPT
SCHEMBL7369952 0.84 ALDH1A1 (0.48) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL9832213 0.81 LTA4H (0.44) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL9832465 0.81 KMT2A (0.49) NPC1RAB9ASMN1; SMN2KMT2AMAPT
SCHEMBL9831766 0.81 TSHR (0.58) NPSR1ALDH1A1KMT2AMAPTHTT
SCHEMBL3982930 0.80 MAPT (0.52) ALDH1A1KMT2AMAPTGAAMEN1
SCHEMBL9830883 0.79 KMT2A (0.44) NPSR1ALDH1A1KMT2AMEN1LMNA
SCHEMBL10845563 0.78 ALDH1A1 (0.69) NPC1RAB9ANPSR1SMN1; SMN2ALDH1A1
SCHEMBL9831436 0.76 TUBB1 (0.51)
SCHEMBL6260691 0.74 RAB9A (0.52) NPC1RAB9ANPSR1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129846-B1 (3-AMINO-1H-PYRAZOL-4-YL)(ARYL)METHANONES AMERICAN CYANAMID COMPANY (US) 1991-05-08 EP claimed
EP-0129846-A2 (3-Amino-1H-pyrazol-4-yl)(aryl)methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP claimed
EP-0129847-A2 Aryl and heteroaryl[7-(aryl and heteroaryl)-pyrazolo-[1,5-a]-pyrimidin-3-yl]methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP disclosed