SCHEMBL9832094

SCHEMBL9832094

O=C1Cc2cc3c(cc2N1)NC(c1cccnc1)N3

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 6/20 0.53
CYP11B2 P19099 6/20 0.53
CYP1A2 P05177 2/20 0.53
MAPT P10636 4/20 0.48
KDM4E B2RXH2 2/20 0.48
MAPK1 P28482 2/20 0.48
MEN1 O00255 1/20 0.48
RECQL P46063 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 1/20 0.48
MCL1 Q07820 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.43
PDE3B Q13370 2/20 0.43
PDE3A Q14432 2/20 0.43
TDP2 O95551 2/20 0.42
CYP19A1 P11511 2/20 0.41
CYP2C9 P11712 1/20 0.40
TBXAS1 P24557 1/20 0.40
TSHR P16473 1/20 0.40
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833717 0.83 PDE3B (0.54) CYP11B1CYP11B2CYP1A2MAPTKDM4E
Hydrochloric Acid SCHEMBL10470469 0.82 PDE3B (0.52) CYP11B1CYP11B2CYP1A2MAPTKDM4E
SCHEMBL10695340 0.76 KDM4E (0.45) CYP11B1CYP11B2CYP1A2MAPTKDM4E
SCHEMBL10698957 0.72 CYP1A2 (0.44) CYP11B1CYP11B2CYP1A2MAPTKDM4E
SCHEMBL10566220 0.72 ALDH1A1 (0.50) MAPTKDM4EMAPK1MEN1KMT2A
SCHEMBL9831252 0.72 KDM4E (0.46) MAPTKDM4EMAPK1MEN1RECQL
SCHEMBL10698931 0.72 KDM4E (0.41) MAPTKDM4EMAPK1MEN1RECQL
SCHEMBL10558735 0.71 MAPT (0.48) MAPTKDM4EMAPK1MEN1RECQL
SCHEMBL1875587 0.70 CYP11B1 (0.78) CYP11B1CYP11B2CYP1A2PDE3BPDE3A
SCHEMBL9831225 0.70 KDM4E (0.44) CYP1A2MAPTKDM4EMAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed
EP-0161632-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1985-11-21 EP disclosed