SCHEMBL10698957

SCHEMBL10698957

CCN1C(=O)Cc2cc3c(cc21)NC(c1cccnc1)N3

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
HTT P42858 1/20 0.43
KDM4E B2RXH2 5/20 0.41
MAPT P10636 4/20 0.41
MEN1 O00255 2/20 0.41
MAPK1 P28482 2/20 0.41
KMT2A Q03164 2/20 0.41
RAB9A P51151 2/20 0.41
RECQL P46063 1/20 0.41
MCL1 Q07820 1/20 0.41
TSHR P16473 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
CYP3A4 P08684 2/20 0.40
THRB P10828 1/20 0.40
THPO P40225 1/20 0.40
POLB P06746 1/20 0.38
BMPR1B O00238 1/20 0.38
BMPR1A P36894 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698931 0.88 KDM4E (0.41) HTTKDM4EMAPTMEN1MAPK1
SCHEMBL10698178 0.86 ALDH1A1 (0.40) CYP1A2CYP11B1CYP11B2HTTKDM4E
SCHEMBL10695340 0.86 KDM4E (0.45) CYP1A2CYP11B1CYP11B2KDM4EMAPT
SCHEMBL10698582 0.85 CYP1A2 (0.41) CYP1A2CYP11B1CYP11B2HTTKDM4E
SCHEMBL10699435 0.79 KMT2A (0.40) HTTMEN1KMT2ABMPR1BBMPR1A
SCHEMBL10699328 0.78 KDM4E (0.41) CYP1A2CYP11B1CYP11B2HTTKDM4E
SCHEMBL10700217 0.78 KDM4E (0.41) CYP1A2CYP11B1CYP11B2HTTKDM4E
SCHEMBL10699549 0.76 BMPR1B (0.41) HTTKDM4EMEN1MAPK1KMT2A
SCHEMBL10698133 0.73 BRD4 (0.36) CYP1A2CYP11B1CYP11B2HTTKDM4E
SCHEMBL9832094 0.72 CYP11B1 (0.53) CYP1A2CYP11B1CYP11B2KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed