SCHEMBL9833717

SCHEMBL9833717

O=C1Cc2cc3c(cc2N1)NC(c1ccncc1)N3

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.54
PDE3A Q14432 2/20 0.54
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 2/20 0.47
CYP1A2 P05177 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
EPHX2 P34913 1/20 0.41
AHR P35869 4/20 0.41
CMA1 P23946 2/20 0.41
EIF2AK2 P19525 1/20 0.40
TSHR P16473 2/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
PDK2 Q15119 1/20 0.38
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10470469 0.99 PDE3B (0.52) PDE3BPDE3AKDM4EALDH1A1HSD17B10
SCHEMBL9832094 0.83 CYP11B1 (0.53) PDE3BPDE3AKDM4EALDH1A1CYP1A2
SCHEMBL9834566 0.76 AHR (0.44) PDE3BPDE3AEPHX2AHRCMA1
SCHEMBL10566220 0.73 ALDH1A1 (0.50) PDE3BPDE3AKDM4EALDH1A1HSD17B10
SCHEMBL31010750 0.73 AHR (0.59) PDE3BPDE3ACYP1A2CYP11B1CYP11B2
SCHEMBL9832061 0.71 PDE3B (0.49) PDE3BPDE3AKDM4EALDH1A1HSD17B10
SCHEMBL23143482 0.70 PDE3B (1.00) PDE3BPDE3ACYP1A2CYP11B1CYP11B2
SCHEMBL6744175 0.70 PDE3B (0.76) PDE3BPDE3ACYP1A2CYP11B1CYP11B2
SCHEMBL29850050 0.70 PDE3B (0.76) PDE3BPDE3ACYP1A2CYP11B1CYP11B2
SCHEMBL9762771 0.70 AHR (0.48) PDE3BPDE3ACYP1A2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed
EP-0161632-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1985-11-21 EP disclosed