SCHEMBL10695340

SCHEMBL10695340

CN1C(=O)Cc2cc3c(cc21)NC(c1cccnc1)N3

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.45
MEN1 O00255 2/20 0.45
MAPK1 P28482 2/20 0.45
KMT2A Q03164 2/20 0.45
MAPT P10636 2/20 0.45
RAB9A P51151 2/20 0.45
RECQL P46063 1/20 0.45
MCL1 Q07820 1/20 0.45
CYP3A4 P08684 3/20 0.43
TSHR P16473 2/20 0.43
THRB P10828 1/20 0.43
THPO P40225 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CYP11B1 P15538 5/20 0.42
CYP11B2 P19099 5/20 0.42
CYP19A1 P11511 4/20 0.42
CYP17A1 P05093 1/20 0.42
CYP1A2 P05177 1/20 0.42
ALDH1A1 P00352 1/20 0.38
BMPR1B O00238 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10698957 0.86 CYP1A2 (0.44) KDM4EMEN1MAPK1KMT2AMAPT
SCHEMBL10694302 0.84 KDM4E (0.43) KDM4EMEN1MAPK1KMT2ACYP3A4
SCHEMBL10698931 0.83 KDM4E (0.41) KDM4EMEN1MAPK1KMT2AMAPT
SCHEMBL9832094 0.76 CYP11B1 (0.53) KDM4EMEN1MAPK1KMT2AMAPT
SCHEMBL10691679 0.76 KDM4E (0.45) KDM4EMEN1MAPK1KMT2AMAPT
SCHEMBL10695479 0.76 KDM4E (0.45) KDM4EMEN1MAPK1KMT2AMAPT
SCHEMBL10698582 0.71 CYP1A2 (0.41) KDM4EMEN1MAPK1KMT2AMAPT
SCHEMBL10695102 0.71 KDM4E (0.38) KDM4ECYP3A4ALDH1A1BMPR1BBMPR1A
SCHEMBL10698178 0.71 ALDH1A1 (0.40) KDM4EKMT2ATSHRCYP11B1CYP11B2
SCHEMBL769062 0.70 CYP11B1 (0.78) CYP3A4CYP11B1CYP11B2CYP19A1CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed