SCHEMBL9833512

SCHEMBL9833512

CCC1(CC)C(=O)Nc2cc3[nH]c(C(C)c4ccncc4)nc3cc21

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
AAK1 Q2M2I8 8/20 0.36
ALDH1A1 P00352 2/20 0.35
PGR P06401 2/20 0.34
KDM4E B2RXH2 2/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
GSK3B P49841 1/20 0.30
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832933 0.80 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9833519 0.77 ALDH1A1 (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9833966 0.75 MAPT (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10472429 0.73 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9832117 0.72 MAPT (0.54) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10373500 0.71 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834616 0.69 PDE3B (0.47) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10553987 0.68 LMNA (0.45) PDE3BPDE3AAAK1PGRKDM4E
SCHEMBL10568502 0.68 ALOX5 (0.47) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10374713 0.68 FBP1 (0.49) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed