SCHEMBL9834705

SCHEMBL9834705

CCCC1C(=O)Nc2cc3c(cc21)NC(O)N3

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 3/20 0.39
IDO1 P14902 1/20 0.36
MAPT P10636 6/20 0.36
GAA P10253 2/20 0.36
PGR P06401 1/20 0.35
TP53 P04637 6/20 0.35
POLB P06746 1/20 0.35
LMNA P02545 4/20 0.34
DRD2 P14416 2/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
PKM P14618 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR7 P34969 2/20 0.33
DRD1 P21728 1/20 0.32
HTR2A P28223 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9834604 0.87 PGR (0.46) NQO2IDO1MAPTGAAPGR
SCHEMBL9834779 0.78 PGR (0.47) NQO2IDO1MAPTPGRTP53
SCHEMBL10470471 0.78 IDO1 (0.41) NQO2IDO1MAPTGAAPGR
SCHEMBL9834389 0.77 PGR (0.41) PGR
SCHEMBL9834101 0.73 MAOB (0.38) IDO1MAPTTP53LMNA
SCHEMBL9833078 0.73 TDP2 (0.49) MAPTGAATP53POLBLMNA
SCHEMBL9835252 0.72 PGR (0.40) NQO2IDO1MAPTGAAPGR
SCHEMBL14996404 0.72 HTR7 (0.54) NQO2IDO1MAPTPGRTP53
SCHEMBL9835010 0.72 PGR (0.44) NQO2IDO1MAPTGAAPGR
SCHEMBL9773669 0.72 POLB (0.48) NQO2IDO1MAPTGAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214592-B1 PYRROLOBENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE PRODUCTS Roche Diagnostics GmbH (DE) 1991-08-14 EP disclosed
US-4730003-A Tricyclic compounds for treating heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-03-08 US disclosed
EP-0214592-A2 Pyrrolobenzimidazoles, process for their preparation and medicaments containing these products Roche Diagnostics GmbH (DE) 1987-03-18 EP disclosed