SCHEMBL9835129

SCHEMBL9835129

COc1cc(OC)c(CC=O)c(O)c1C

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.49
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
FASN P49327 1/20 0.42
ERN1 O75460 4/20 0.41
IMPDH2 P12268 2/20 0.38
ABCB1 P08183 5/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13450126 0.84 IMPDH2 (0.41) CYP3A4MEN1KMT2ARXFP1FASN
SCHEMBL16166121 0.83 ABCB1 (0.46) CYP3A4FASNERN1ABCB1TDP1
SCHEMBL8699353 0.76 ERN1 (0.47) MEN1KMT2ARXFP1ERN1IMPDH2
SCHEMBL8571840 0.74 FASN (0.48) CYP3A4MEN1KMT2ARXFP1FASN
SCHEMBL743276 0.72 ERN1 (0.57) CYP3A4KMT2AERN1
SCHEMBL29694978 0.72 ERN1 (0.47) CYP3A4ERN1ALDH1A1
SCHEMBL4054977 0.72 MAPT (0.51) CYP3A4KMT2AERN1KDM4E
SCHEMBL14262143 0.71 TNKS2 (0.47) CYP3A4ERN1ALDH1A1
SCHEMBL15266045 0.71 ALOX5 (0.44) ERN1IMPDH2
SCHEMBL21626905 0.71 ALDH1A1 (0.41) CYP3A4MEN1KMT2ARXFP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415566-A1 Heterocyclic compounds, processes for producing them and pharmaceutical compositions comprising them SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1991-03-06 EP disclosed