SCHEMBL9835781

SCHEMBL9835781

CCN1C(=O)C2=C(c3cccc(Cl)c3)N(CC)C(=O)C2=C1c1cccc(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.46
NR1H3 Q13133 2/20 0.46
PGR P06401 4/20 0.45
ALDH1A1 P00352 5/20 0.40
POLB P06746 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
KDM4E B2RXH2 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 1/20 0.38
BACE1 P56817 2/20 0.38
CTSD P07339 1/20 0.38
TAAR1 Q96RJ0 2/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837963 0.80 NR1H2 (0.50) NR1H2NR1H3ALDH1A1APOBEC3GKDM4E
SCHEMBL9835835 0.79 NR1H2 (0.56) NR1H2NR1H3ALDH1A1KDM4EKMT2A
SCHEMBL9834685 0.78 PGR (0.51) PGRALDH1A1POLBKDM4EKMT2A
SCHEMBL7504411 0.75 GAA (0.42) PGRALDH1A1KDM4EKMT2AMEN1
SCHEMBL8069949 0.70 XPO1 (0.43) PGRKMT2AMEN1
SCHEMBL15353831 0.70 NR1H2 (0.47) NR1H2NR1H3ALDH1A1HSD17B10KMT2A
SCHEMBL16456162 0.69 SENP1 (0.39) NR1H2NR1H3ALDH1A1LMNANPSR1
SCHEMBL10050134 0.69 NR1H2 (0.46) NR1H2NR1H3ALDH1A1KDM4ECYP1A2
SCHEMBL4685918 0.68 NR1H2 (0.60) NR1H2NR1H3ALDH1A1KDM4ELMNA
SCHEMBL18327868 0.68 NR1H2 (0.44) NR1H2NR1H3ALDH1A1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0133156-B1 1,4-DIKETOPYRROLO-(3,4-C) PYRROLES CIBA-GEIGY AG (CH) 1991-07-10 EP disclosed
US-4666455-A Compositions pigmented with N-substituted 1,4-diketopyrrolo-[3,4-c]-pyrroles CIBA-GEIGY CORPORATION (US) 1987-05-19 US disclosed
US-4585878-A N-substituted 1,4-diketopyrrolo-[3,4-c]-pyrroles CIBA-GEIGY CORPORATION (US) 1986-04-29 US disclosed
EP-0133156-A2 1,4-Diketopyrrolo-(3,4-c) pyrroles CIBA-GEIGY AG (CH) 1985-02-13 EP disclosed