SCHEMBL9834685

SCHEMBL9834685

CN1C(=O)C2=C(c3cccc(Cl)c3)N(C)C(=O)C2=C1c1cccc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PGR P06401 6/20 0.51
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MAOB P27338 2/20 0.43
MAOA P21397 1/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
BACE1 P56817 1/20 0.43
IDO1 P14902 1/20 0.42
ESR2 Q92731 1/20 0.42
ALOX5 P09917 1/20 0.42
TGFBR1 P36897 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837439 0.80 RAB9A (0.41) PGRMAPTKMT2ATGFBR1
SCHEMBL7068310 0.79 PTGS2 (0.51) ALDH1A1MEN1MAPTHPGDKMT2A
SCHEMBL7504411 0.79 GAA (0.42) PGRALDH1A1MEN1MAPTKMT2A
SCHEMBL14479768 0.79 NR1H2 (0.37) PGRALDH1A1MEN1POLBKMT2A
SCHEMBL9835781 0.78 NR1H2 (0.46) PGRALDH1A1MEN1POLBKMT2A
SCHEMBL5070001 0.77 NR1H2 (0.52) MAPTTDP1GAA
SCHEMBL12725181 0.75 NR1H2 (0.50) ALDH1A1MAPT
SCHEMBL9836649 0.75 PGR (0.46) PGRBACE1TGFBR1
SCHEMBL14620062 0.73 COMT (0.40) ALDH1A1MEN1MAPTKMT2AMAOB
SCHEMBL6003662 0.72 PGR (0.46) PGRALDH1A1MEN1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0133156-B1 1,4-DIKETOPYRROLO-(3,4-C) PYRROLES CIBA-GEIGY AG (CH) 1991-07-10 EP disclosed
US-4666455-A Compositions pigmented with N-substituted 1,4-diketopyrrolo-[3,4-c]-pyrroles CIBA-GEIGY CORPORATION (US) 1987-05-19 US disclosed
US-4585878-A N-substituted 1,4-diketopyrrolo-[3,4-c]-pyrroles CIBA-GEIGY CORPORATION (US) 1986-04-29 US disclosed