SCHEMBL9836255

SCHEMBL9836255

O=C(Cl)c1cccc(F)c1C(=O)Cl

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.65
ALOX15 P16050 1/20 0.65
CES2 O00748 4/20 0.54
CES1 P23141 4/20 0.54
BCHE P06276 1/20 0.48
ALB P02768 1/20 0.45
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
LMNA P02545 2/20 0.41
GAA P10253 2/20 0.40
TDP1 Q9NUW8 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL105255 0.86 CES2 (0.64) ALDH1A1ALOX15CES2CES1BCHE
SCHEMBL8702458 0.86 CES2 (0.59) ALDH1A1ALOX15CES2CES1BCHE
SCHEMBL15578239 0.84 CES2 (0.61) ALDH1A1ALOX15CES2CES1BCHE
SCHEMBL893277 0.84 ALDH1A1 (0.56) ALDH1A1ALOX15CES2CES1BCHE
SCHEMBL27900422 0.83 ALDH1A1 (0.60) ALDH1A1ALOX15CES2CES1BCHE
SCHEMBL853194 0.81 ALDH1A1 (0.53) ALDH1A1ALOX15CES2CES1KMT2A
SCHEMBL104744 0.80 CES2 (0.68) ALDH1A1ALOX15CES2CES1BCHE
Methylene Chloride SCHEMBL28186741 0.80 CES2 (0.56) ALDH1A1ALOX15CES2CES1BCHE
SCHEMBL30733529 0.79 ALDH1A1 (1.00) ALDH1A1ALOX15CES2CES1BCHE
SCHEMBL60101 0.79 ALDH1A1 (1.00) ALDH1A1ALOX15CES2CES1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0253837-B1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS MALLINCKRODT SPECIALTY CHEMICALS COMPANY (US) 1991-10-09 EP disclosed
EP-0252964-B1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS MALLINCKRODT SPECIALTY CHEMICALS COMPANY (US) 1991-08-21 EP disclosed
EP-0253838-B1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING N-SEC-ALKYL PYRIDINIUM SALTS MALLINCKRODT SPECIALTY CHEMICALS COMPANY (US) 1991-08-21 EP disclosed
US-4973771-A Phase transfer catalysts MALLINCKRODT, INC. (US) 1990-11-27 US disclosed
US-4973772-A Catalytic method for producing fluoroarmatic compounds using substituted pyridinium salts MALLINCKRODT, INC. (US) 1990-11-27 US disclosed
EP-0253836-B1 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE Mallinckrodt, Inc. (a Delaware corporation) (US) 1990-10-03 EP disclosed
US-4927980-A REACTING CHLOROAROMATIC COMPOUND WITH ALKALI METAL FLUORIDE SALTS MALLINCKRODT INC. (US) 1990-05-22 US disclosed
US-4849552-A METHANOL, AROMATIC HYDROCARBON OR HALOCARBON, AZEOTROPES MALLINCKRODT, INC. (US) 1989-07-18 US disclosed
EP-0252964-A4 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-07-14 EP disclosed
EP-0253836-A4 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE. MALLINCKRODT INC (US) 1988-04-27 EP disclosed
EP-0253837-A4 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-04-26 EP disclosed
EP-0253836-A1 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE. MALLINCKRODT INC (US) 1988-01-27 EP disclosed
EP-0253837-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-01-27 EP disclosed
EP-0252964-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-01-20 EP disclosed
WO-1987004148-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS MALLINCKRODT, INC. (US) 1987-07-16 WO disclosed
WO-1987004149-A1 PHASE TRANSFER CATALYSTS MALLINCKRODT, INC. (US) 1987-07-16 WO disclosed
WO-1987004151-A1 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE MALLINCKRODT, INC. (US) 1987-07-16 WO disclosed
WO-1987004150-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS MALLINCKRODT, INC. (US) 1987-07-16 WO disclosed