SCHEMBL9837076

SCHEMBL9837076

COC(=O)C1=C(C)N(c2ccccc2C)C(C)=C(C(=O)OC)C1c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.64
TSHR P16473 4/20 0.52
GAA P10253 2/20 0.52
HSD17B10 Q99714 3/20 0.50
KDM4E B2RXH2 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
ADORA3 P0DMS8 1/20 0.49
HPGD P15428 1/20 0.49
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 5/20 0.45
LMNA P02545 2/20 0.45
RECQL P46063 1/20 0.45
CACNA1F O60840 1/20 0.45
CACNA1D Q01668 1/20 0.45
CACNA1S Q13698 1/20 0.45
CACNA1C Q13936 1/20 0.45
HTT P42858 2/20 0.44
CASP1 P29466 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836397 0.85 NOTUM (0.45) POLBTSHRGAAKDM4EKMT2A
SCHEMBL5363492 0.80 TSHR (0.74) POLBTSHRGAAHSD17B10KDM4E
SCHEMBL11863359 0.75 TSHR (0.67) POLBTSHRGAAHSD17B10KDM4E
SCHEMBL9033145 0.72 POLB (0.54) POLBTSHRGAAHSD17B10KDM4E
SCHEMBL3905675 0.72 ADORA3 (0.83) POLBTSHRGAAHSD17B10KDM4E
SCHEMBL7920096 0.72 ALDH1A1 (0.66) POLBTSHRHSD17B10ADORA3KMT2A
SCHEMBL9836195 0.70 LMNA (0.53) POLBTSHRGAAHSD17B10KDM4E
SCHEMBL10517002 0.70 LMNA (0.53) POLBTSHRGAAHSD17B10KDM4E
SCHEMBL7266889 0.69 POLB (0.51) POLBTSHRGAAHSD17B10KDM4E
SCHEMBL6951320 0.69 ADORA3 (0.76) POLBTSHRGAAHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0234776-B1 PROCESS FOR 1,4-DIHYDROPYRIDINE COMPOUNDS MERCK & CO. INC. (US) 1991-09-04 EP disclosed
US-4780538-A REACTING AN AMINOALKENOATE WITH AN AROMATIC ALDEHYDE USING AN TITANAMINE CATALYST MERCK & CO., INC. (US) 1988-10-25 US disclosed
EP-0234776-A2 Process for 1,4-dihydropyridine compounds MERCK & CO. INC. (US) 1987-09-02 EP disclosed