SCHEMBL9836779

SCHEMBL9836779

COC(=O)C1=Cc2sc(Cn3ccnc3)cc2CC1

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 16/20 0.76
KDM4E B2RXH2 1/20 0.36
AHR P35869 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CYP19A1 P11511 1/20 0.36
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835184 0.89 TBXAS1 (0.61) TBXAS1KDM4EAHRNPSR1
Imitrodast SCHEMBL166460 0.86 TBXAS1 (1.00) TBXAS1
Imitrodast SCHEMBL8156405 0.85 TBXAS1 (0.81) TBXAS1KDM4ECYP19A1
Imitrodast SCHEMBL99497 0.85 TBXAS1 (0.98) TBXAS1
SCHEMBL9835177 0.83 TBXAS1 (0.53) TBXAS1KDM4EAHRNPSR1CYP19A1
SCHEMBL9835676 0.83 TBXAS1 (0.76) TBXAS1KDM4EAHRNPSR1CYP19A1
SCHEMBL9836523 0.81 TBXAS1 (0.74) TBXAS1
SCHEMBL9401600 0.79 TBXAS1 (0.67) TBXAS1KDM4ECYP19A1
SCHEMBL9835663 0.78 TBXAS1 (0.43) TBXAS1KDM4ENPC1
SCHEMBL9836683 0.78 TBXAS1 (0.52) TBXAS1KDM4EAHRNPSR1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-62252784-A None JP disclosed
EP-0240107-B1 THIANAPHTHENE DERIVATIVES, THEIR PRODUCTION AND USE Sankyo Company Limited (JP) 1991-08-21 EP disclosed
US-5021444-A Anticoagulants SANKYO COMPANY LIMITED (JP) 1991-06-04 US disclosed
US-4847272-A ANTICOAGULANTS SANKYO COMPANY LIMITED (JP) 1989-07-11 US disclosed
JP-S62252784-A THIANAPHTHENE DERIVATIVE AND PRODUCTION THEREOF SANKYO CO LTD 1987-11-04 JP disclosed
EP-0240107-A1 Thianaphthene derivatives, their production and use Sankyo Company Limited (JP) 1987-10-07 EP disclosed