SCHEMBL9837007

SCHEMBL9837007

O=C1c2ccccc2C(=O)N1C/C=C/CN1CCN(C(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.67
DRD3 P35462 6/20 0.67
GAA P10253 3/20 0.64
NPSR1 Q6W5P4 3/20 0.64
ALDH1A1 P00352 2/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
POLB P06746 1/20 0.64
LMNA P02545 4/20 0.62
HIF1A Q16665 4/20 0.62
CYP3A4 P08684 3/20 0.62
CYP2D6 P10635 3/20 0.62
OPRD1 P41143 3/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2C9 P11712 2/20 0.62
CHRM2 P08172 2/20 0.62
CHRM4 P08173 2/20 0.62
HTR1A P08908 2/20 0.62
CHRM5 P08912 2/20 0.62
ADRA2A P08913 2/20 0.62
ADORA3 P0DMS8 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837012 1.00 DRD2 (0.67) DRD2DRD3GAANPSR1ALDH1A1
SCHEMBL9733689 0.83 DRD2 (0.84) DRD2DRD3GAANPSR1ALDH1A1
SCHEMBL31232750 0.83 DRD2 (0.84) DRD2DRD3GAANPSR1ALDH1A1
SCHEMBL9256633 0.81 DRD2 (1.00) DRD2DRD3GAANPSR1ALDH1A1
SCHEMBL7976323 0.81 DRD2 (0.95) DRD2DRD3GAANPSR1ALDH1A1
SCHEMBL1137893 0.80 OPRD1 (0.68) DRD2DRD3GAANPSR1ALDH1A1
SCHEMBL9837345 0.80 OPRD1 (0.68) DRD2DRD3GAANPSR1ALDH1A1
SCHEMBL1137896 0.80 OPRD1 (0.68) DRD2DRD3GAANPSR1ALDH1A1
SCHEMBL9837343 0.80 OPRD1 (0.68) DRD2DRD3GAANPSR1ALDH1A1
Hydrochloric Acid SCHEMBL10826808 0.80 DRD2 (0.92) DRD2DRD3GAANPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0210782-B1 PYRIDINE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Dainippon Pharmaceutical Co., Ltd. (JP) 1991-04-17 EP disclosed
US-4778796-A ω-(3-pyridyl)alkenamide derivatives and anti-allergenic pharmaceutical compositions containing same DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1988-10-18 US disclosed
EP-0210782-A2 Pyridine compounds, process for the preparation thereof and pharmaceutical composition containing the same Dainippon Pharmaceutical Co., Ltd. (JP) 1987-02-04 EP disclosed